Target Details
| UniProt AC | P21731 |
|---|---|
| Gene Symbol | TBXA2R |
| Protein Name | Thromboxane A2 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 286
- Clinical molecules 6
- Avg pChEMBL 7.02
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (286)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ISMHAZMNDUAHLK
|
7.8 | IC50 | 2 | — | |
QOIVFTOIMRANMQ
|
7.8 | IC50 | 2 | — | |
QOIVFTOIMRANMQ
|
7.7 | IC50 | 2 | — | |
ZDZJTARQTIAZKQ
|
7.7 | Ki | 2 | — | |
LGHLGTHRJNIRCA
|
7.7 | IC50 | 2 | — | |
NUPJOHLAKYWZHZ
|
7.7 | IC50 | 2 | — | |
IEZMFLQSTWTPEP
|
7.7 | IC50 | 2 | — | |
ANSZFKJHEBXZMZ
|
7.6 | Ki | 2 | — | |
RERMKDAOFJRCJU
|
7.6 | IC50 | 2 | — | |
WBSMJRCXYPFSIK
|
7.6 | Ki | 2 | — | |
GUTGDFJEUBLDBQ
|
7.6 | IC50 | 2 | — | |
SDGUUEATIIAOTG
|
7.6 | Ki | 2 | — | |
JIOGHZHDRQMSBB
|
7.6 | IC50 | 2 | — | |
JIOGHZHDRQMSBB
|
7.6 | IC50 | 2 | — | |
AQQCPDIIPNDMEK
|
7.6 | Kd | 2 | — | |
KVNYICIYEISPHS
|
7.5 | IC50 | 2 | — | |
NMJYFIAGWNELHF
|
7.5 | IC50 | 2 | — | |
UYIFEFLIAAUJOU
|
7.5 | IC50 | 2 | — | |
JLQUGIOTHHQRSB
|
7.5 | IC50 | 2 | — | |
JLQUGIOTHHQRSB
|
7.5 | IC50 | 2 | — | |
FECWOVCONGPURJ
|
7.5 | Ki | 3 | — | |
KEKQERHYRPEXLS
|
7.5 | IC50 | 2 | — | |
SHRNOBNPOTZEAM
|
7.5 | IC50 | 2 | — | |
KEKQERHYRPEXLS
|
7.5 | IC50 | 2 | — | |
UICLKHCKXGFMBB
|
7.5 | Kd | 2 | — | |
WICGPTMBFXQNBE
|
7.5 | IC50 | 2 | — | |
XBMUFQALKMIYCY
|
7.5 | IC50 | 2 | — | |
TXKRKUVUYCOYKP
|
7.5 | IC50 | 2 | — | |
TXKRKUVUYCOYKP
|
7.5 | IC50 | 2 | — | |
AERMYTSNNRHMDS
|
7.4 | IC50 | 2 | — | |
XYLHWYSIVHTCSV
|
7.4 | Ki | 2 | — | |
RGGXEZXJJJANGJ
|
7.4 | IC50 | 2 | — | |
RGGXEZXJJJANGJ
|
7.4 | IC50 | 2 | — | |
FJMQKJOWJVMHPQ
|
7.4 | Ki | 5 | — | |
SSRGVHMXPYHYSL
|
7.4 | Ki | 2 | — | |
CDTZYZWEPCKHSB
|
7.4 | IC50 | 2 | — | |
KDYFIMFGTYIEBR
|
7.4 | Ki | 2 | — | |
SOUOKSHPPGIZRL
|
7.4 | IC50 | 2 | — | |
OICNDPFYFJKIKF
|
7.4 | IC50 | 2 | — | |
WMXZEBHSAJEWND
|
7.4 | Kd | 2 | — | |
SHRNOBNPOTZEAM
|
7.3 | IC50 | 2 | — | |
BRVYETPRGCQZJA
|
7.3 | Ki | 2 | — | |
QGTKGOGDYIAADK
|
7.3 | IC50 | 2 | — | |
QGTKGOGDYIAADK
|
7.3 | IC50 | 2 | — | |
KEOWJWUNPZAGBC
|
7.3 | IC50 | 2 | — | |
HQNOTLSNWDHOJY
|
7.3 | Ki | 3 | — | |
WSGAKKPWXZPETA
|
7.3 | IC50 | 2 | — | |
RROZSWAPBMHDGH
|
7.3 | IC50 | 2 | — | |
UTAFETDONDFNBQ
|
7.3 | Kd | 2 | — | |
LQANGKSBLPMBTJ
|
7.3 | Ki | 3 | — |