Target Details
UniProt ACP21731
Gene SymbolTBXA2R
Protein NameThromboxane A2 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 286
  • Clinical molecules 6
  • Avg pChEMBL 7.02
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (286)
InChIKey pChEMBL Type Targets Clinical
BRIAEVLTRZHLAS 8.8 Ki 2
BTWTZWMDGIJYTQ 8.7 Ki 2
AEIQZZAOZDLCSH 8.6 Ki 2
BBQILAZFNVDEMU 8.6 Kd 2
USPFQIRXYBZUPX 8.6 Ki 2
WPBWMPUZDXLQIX 8.6 Kd 2
CGSLOOCFBLEGKW 8.6 Ki 2
PWTCIBWRMQFJBC 8.5 Kd 2
JEJFHDDECMACOD 8.5 IC50 2
MBFUMLZEULKFON 8.5 IC50 2
LIYMSLCFOJXHRD 8.4 Ki 2
AGAXMMPHPXHEAW 8.4 Kd 2
IDSQFTJASXFWNN 8.4 Kd 2
VGBBXLWOWUXXFE 8.4 Kd 2
VQNGUZVGSDDDEI 8.3 Ki 2
AEMOPCLSCUUOFI 8.3 Kd 2
LOFDECJHZOIDID 8.3 Ki 3
VKYMAXGZPKUBLB 8.2 Kd 2
HSKIZOWUDQCJET 8.2 Ki 2
RCUUGUXXIMFUAQ 8.2 Ki 2
SWLNUQSMWKYMJE 8.2 IC50 2
SWLNUQSMWKYMJE 8.2 IC50 2
XOXVIHCDCWSEJJ 8.1 Ki 2
XSQAICBCYIFUQS 8.1 IC50 5
ASLWQKCVXKAGOH 8.1 IC50 2
YNLWPJVDHZFCOY 8.0 Ki 2
HCLFUHWPLXVRIS 8.0 Kd 2
HJPAXYLYYQIFCK 8.0 Ki 2
ZNRZNAHHOIANAO 8.0 Kd 2
RJNDVCNWVBWHLY 8.0 Ki 2
NXFFJDQHYLNEJK 8.0 IC50 6
XUTLOCQNGLJNSA 8.0 IC50 2
XUTLOCQNGLJNSA 8.0 IC50 2
XUTLOCQNGLJNSA 8.0 IC50 2
CIWXNRVCXQIBPC 7.9 IC50 2
LJZXVXGFHZARCP 7.9 IC50 2
LMSWDFLNAYPJJD 7.9 Kd 2
LQZKCALSANZAMX 7.9 IC50 2
LQZKCALSANZAMX 7.9 IC50 2
YKPJTNNQDJFQBF 7.9 Kd 2
KHQYDHFXPAZDBK 7.9 IC50 2
LZONHUSMVCYUJX 7.9 Ki 2
YYAWOSLKARYYMV 7.8 Ki 3
LTCQRNQPODCPAS 7.8 Kd 2
LTCQRNQPODCPAS 7.8 Kd 2
XYEOSUOFNKZBKV 7.8 IC50 2
XYEOSUOFNKZBKV 7.8 IC50 2
GSBAVONRPNJJOH 7.8 Ki 2
IMMNAXXZSBKGMT 7.8 IC50 2
IMMNAXXZSBKGMT 7.8 IC50 2
2D structure