Target Details
| UniProt AC | P21730 |
|---|---|
| Gene Symbol | C5AR1 |
| Protein Name | C5a anaphylatoxin chemotactic receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 5
- Clinical molecules 0
- Avg pChEMBL 7.01
KEGG Pathways (6)
Active Molecules (5)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YOKBGCTZYPOSQM
|
7.5 | IC50 | 4 | — | |
HXKFHHNEFCZKPG
|
7.4 | IC50 | 3 | — | |
KPJVSWMSLFZHBU
|
6.9 | Kd | 3 | — | |
KPJVSWMSLFZHBU
|
6.9 | Kd | 3 | — | |
CYLQZMDPLMYAJE
|
6.2 | IC50 | 2 | — |