Target Details
| UniProt AC | P21728 |
|---|---|
| Gene Symbol | DRD1 |
| Protein Name | D(1A) dopamine receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 738
- Clinical molecules 30
- Avg pChEMBL 7.2
KEGG Pathways (12)
Active Molecules (738)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UENAJMHEKJGFHA
|
7.1 | Ki | 2 | — | |
ITGZZZYNPULRNZ
|
7.1 | IC50 | 2 | — | |
JNNOSTQEZICQQP
|
7.1 | Ki | 7 | — | |
KVOKGAUQGXOEAL
|
7.1 | IC50 | 2 | — | |
QAFWRHMUHQYYGU
|
7.1 | Ki | 2 | — | |
ZSTKHSQDNIGFLM
|
7.1 | Ki | 22 | — | |
LNEPOXFFQSENCJ
|
7.1 | Ki | 33 | Yes | |
QGAZPZGGCFPPIQ
|
7.1 | IC50 | 2 | — | |
SDOMGHNXSMDPGR
|
7.1 | IC50 | 2 | — | |
BHUNVFVEHNURLZ
|
7.1 | Ki | 4 | — | |
RHPCETHLGGFAQB
|
7.1 | Ki | 9 | — | |
USBUDHMXOXUPOI
|
7.1 | IC50 | 2 | — | |
VIVYNGHHCGDRHE
|
7.1 | IC50 | 2 | — | |
LHHCQDFZJQYUSF
|
7.1 | Ki | 2 | — | |
BFYNQIVBIQGLJA
|
7.1 | Ki | 2 | — | |
FDMHBTAXJFCYLV
|
7.1 | IC50 | 2 | — | |
FJUALPUCFNOCDA
|
7.1 | Ki | 2 | — | |
QGAZPZGGCFPPIQ
|
7.1 | IC50 | 2 | — | |
QMEAXKMTOSHGKG
|
7.1 | Ki | 2 | — | |
ASMVKSNPCVNVFO
|
7.0 | Ki | 5 | — | |
INRYDSYGYMQFRB
|
7.0 | Ki | 5 | — | |
IWMPNKVRIUOVNY
|
7.0 | Ki | 2 | — | |
QZUDBNBUXVUHMW
|
7.0 | Ki | 39 | Yes | |
RMKVCRINIVDQQR
|
7.0 | Ki | 2 | — | |
DXEOLSCGMKPOSP
|
7.0 | IC50 | 2 | — | |
FJIQRQMSPDCJJA
|
7.0 | IC50 | 2 | — | |
ZHWINCTXRNCCKY
|
7.0 | Ki | 2 | — | |
ZPEIMTDSQAKGNT
|
7.0 | Ki | 35 | Yes | |
XODYFOOKKAGIOI
|
7.0 | Ki | 2 | — | |
AYDICYGRWUFLHA
|
7.0 | Ki | 2 | — | |
BEKOHGQOLPINNR
|
7.0 | IC50 | 2 | — | |
KLBQZWRITKRQQV
|
7.0 | Ki | 21 | — | |
NEQWPVBUZDJIHK
|
7.0 | IC50 | 2 | — | |
YOOBJJUPLPSYTE
|
7.0 | IC50 | 2 | — | |
BGGURFWLEHSLEY
|
7.0 | IC50 | 2 | — | |
HFQACMCWJYLKKX
|
7.0 | IC50 | 2 | — | |
YHPPFQXIQZIMOW
|
7.0 | Ki | 5 | — | |
ILRFVZOWNPFKOR
|
7.0 | Ki | 5 | — | |
JVNZVNCHIUVRJV
|
7.0 | IC50 | 2 | — | |
MMSWJNGRQBXTAK
|
7.0 | IC50 | 2 | — | |
WIKYUJGCLQQFNW
|
7.0 | IC50 | 23 | Yes | |
WPJSNLWFVMFFSG
|
7.0 | Ki | 4 | — | |
XASNYJJSDRRREO
|
7.0 | IC50 | 2 | — | |
XEJNCXFNKSUHHY
|
7.0 | Ki | 5 | — | |
AOWOZJJGVFTXQU
|
7.0 | IC50 | 2 | — | |
JJCFRYNCJDLXIK
|
7.0 | IC50 | 25 | Yes | |
SECXHJRGBAZUCO
|
7.0 | Ki | 4 | — | |
DCBIJCAUUCDMMT
|
6.9 | IC50 | 2 | — | |
AYFAGRAOJPSHSH
|
6.9 | Ki | 19 | — | |
DXEOLSCGMKPOSP
|
6.9 | IC50 | 2 | — |