Target Details
| UniProt AC | P21709 |
|---|---|
| Gene Symbol | EPHA1 |
| Protein Name | Ephrin type-A receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 44
- Clinical molecules 11
- Avg pChEMBL 7.02
KEGG Pathways (1)
Active Molecules (44)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JTWMOWRMSZZHDR
|
8.5 | IC50 | 13 | — | |
ZBNZXTGUTAYRHI
|
8.4 | Kd | 102 | Yes | |
ALKJNCZNEOTEMP
|
8.3 | Kd | 55 | — | |
SFCBIFOAGRZJNX
|
8.3 | Kd | 22 | — | |
CXQHYVUVSFXTMY
|
8.2 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
8.2 | Kd | 149 | — | |
VAARYSWULJUGST
|
8.2 | Kd | 119 | Yes | |
FNHKPVJBJVTLMP
|
8.2 | Kd | 29 | — | |
HVXKQKFEHMGHSL
|
8.1 | Kd | 21 | — | |
CIGMIXWAESLRNR
|
8.0 | Kd | 5 | — | |
OUKYUETWWIPKQR
|
8.0 | Kd | 31 | Yes | |
DFJSJLGUIXFDJP
|
7.8 | Kd | 9 | — | |
MJHOMTRKVMKCNE
|
7.5 | IC50 | 12 | — | |
QQWUGDVOUVUTOY
|
7.4 | Kd | 231 | Yes | |
NHHQJBCNYHBUSI
|
7.2 | Kd | 220 | — | |
DKZYXHCYPUVGAF
|
7.0 | Kd | 112 | — | |
JCJSAFZMXVQVBR
|
7.0 | IC50 | 11 | Yes | |
MFAQYJIYDMLAIM
|
7.0 | Kd | 130 | Yes | |
MIMOHMCANSGXIG
|
7.0 | IC50 | 15 | — | |
HKSZLNNOFSGOKW
|
6.9 | IC50 | 408 | — | |
KTEIFNKAUNYNJU
|
6.8 | Kd | 114 | — | |
PHXJVRSECIGDHY
|
6.8 | IC50 | 59 | — | |
VCZDFACOFNRTMG
|
6.8 | IC50 | 6 | — | |
WVXNSAVVKYZVOE
|
6.8 | IC50 | 92 | — | |
YYLKKYCXAOBSRM
|
6.8 | Kd | 191 | — | |
KDGFLJKFZUIJMX
|
6.7 | Kd | 10 | — | |
UHTHHESEBZOYNR
|
6.6 | Kd | 66 | Yes | |
LVLFSSZNAIKYCD
|
6.5 | IC50 | 19 | — | |
HKSZLNNOFSGOKW
|
6.5 | Kd | 213 | — | |
ZCCPLJOKGAACRT
|
6.5 | IC50 | 599 | — | |
ZFKQQXLECNVLOF
|
6.5 | IC50 | 7 | — | |
UIARLYUEJFELEN
|
6.4 | Kd | 289 | Yes | |
LSEAQLOYCHTEOK
|
6.4 | IC50 | 10 | — | |
HHZIURLSWUIHRB
|
6.2 | Kd | 57 | Yes | |
NXSJMRCTGYTSTK
|
6.2 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
6.2 | Kd | 170 | — | |
MVCOAUNKQVWQHZ
|
6.2 | IC50 | 54 | Yes | |
ULTCRVJUAZCGPP
|
6.2 | IC50 | 5 | — | |
BFSMGDJOXZAERB
|
6.2 | Kd | 33 | — | |
JOOXLOJCABQBSG
|
6.1 | Kd | 139 | — | |
GCIKSSRWRFVXBI
|
6.0 | Kd | 109 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |