Target Details
| UniProt AC | P21675 |
|---|---|
| Gene Symbol | TAF1 |
| Protein Name | Transcription initiation factor TFIID subunit 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF12157 (DUF3591) PF09247 (TBP-binding) PF15288 (zf-CCHC_6) |
Summary
- Multi-target molecules 93
- Clinical molecules 0
- Avg pChEMBL 7.35
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (93)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YKDUUWMPYBJPOG
|
7.3 | IC50 | 2 | — | |
NZCCNFWSBAAKSI
|
7.3 | IC50 | 3 | — | |
XWUSNMULJMQCCC
|
7.2 | IC50 | 3 | — | |
YHMNROQTPUKNLA
|
7.2 | IC50 | 8 | — | |
WNTOXMAGPDYDCR
|
7.2 | IC50 | 3 | — | |
SDVGDLDABOUUIN
|
7.2 | IC50 | 2 | — | |
YFDCRPUOAPKOIE
|
7.1 | IC50 | 2 | — | |
BIWUSHWRFMMMGV
|
7.1 | IC50 | 2 | — | |
JJGHZALDUUMGCU
|
7.1 | IC50 | 3 | — | |
WVPDDEACKJQZHD
|
7.1 | IC50 | 2 | — | |
AGCMTUNUCHFYSQ
|
7.0 | IC50 | 2 | — | |
AMEZIZUFNQNCRU
|
7.0 | IC50 | 2 | — | |
CMTGUEFAXALUTH
|
7.0 | IC50 | 3 | — | |
WDUULYPCWOELII
|
7.0 | IC50 | 2 | — | |
OTKIKJDBYKBEOE
|
7.0 | IC50 | 3 | — | |
RBUYFHLQNPJMQM
|
7.0 | Kd | 10 | — | |
KPWWFNXRLAAREN
|
7.0 | Kd | 12 | — | |
XQSKFZQVORBNFZ
|
7.0 | IC50 | 2 | — | |
MOIBHLHUAXJLCW
|
6.8 | IC50 | 5 | — | |
NGXAMXNWIHBLBN
|
6.8 | Kd | 6 | — | |
XQVVPGYIWAGRNI
|
6.8 | IC50 | 34 | — | |
MCVXORPOSRGRKJ
|
6.7 | IC50 | 2 | — | |
QFRIGJQJVRCBFQ
|
6.7 | IC50 | 3 | — | |
XYWMSJMLQUWWJF
|
6.6 | IC50 | 2 | — | |
OHUHVTCQTUDPIJ
|
6.6 | Kd | 4 | — | |
GJAOBHJPGJZEDC
|
6.5 | IC50 | 2 | — | |
JCGPEZVAHLBGMA
|
6.5 | IC50 | 2 | — | |
JGOZUFGBTSAWEI
|
6.5 | Kd | 4 | — | |
UVLQPEQLDXIGTF
|
6.5 | IC50 | 2 | — | |
GAKSHNAOHQIPHD
|
6.5 | IC50 | 2 | — | |
WZQLVEPIBAOOGF
|
6.4 | Kd | 9 | — | |
KHVSTZSCKUIMFH
|
6.4 | IC50 | 3 | — | |
RJEMCUZKQLRUIS
|
6.4 | IC50 | 4 | — | |
OHUHVTCQTUDPIJ
|
6.4 | IC50 | 2 | — | |
AEFZUARQXKQPMD
|
6.3 | IC50 | 2 | — | |
DBLNLPCEKQBLAI
|
6.3 | IC50 | 3 | — | |
BQAKOVGAYWUDIT
|
6.3 | IC50 | 3 | — | |
YXPVTKHEWGXKEY
|
6.2 | Kd | 2 | — | |
UFJLBLXSGFZNIM
|
6.2 | IC50 | 2 | — | |
ZKIRTFGYQVXNGL
|
6.2 | Kd | 2 | — | |
ZKBQMZPFWKZUJV
|
6.1 | IC50 | 2 | — | |
POICMTYCJMMADL
|
6.1 | IC50 | 3 | — | |
SPSRAFOXVSNAJA
|
6.1 | IC50 | 3 | — |