Target Details
| UniProt AC | P21675 |
|---|---|
| Gene Symbol | TAF1 |
| Protein Name | Transcription initiation factor TFIID subunit 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF12157 (DUF3591) PF09247 (TBP-binding) PF15288 (zf-CCHC_6) |
Summary
- Multi-target molecules 93
- Clinical molecules 0
- Avg pChEMBL 7.35
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (93)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVVAQGWHNXKWKB
|
9.7 | Ki | 2 | — | |
IUAWXQMTKGNBRT
|
8.9 | Ki | 2 | — | |
NMRMIPFJPBQHHY
|
8.5 | IC50 | 2 | — | |
KWYIXQZKANFDQR
|
8.4 | IC50 | 2 | — | |
OFZUZFZNFMUNAS
|
8.4 | IC50 | 3 | — | |
YDDKRKCQSIKAJD
|
8.4 | IC50 | 3 | — | |
YTQRBAXLTKDECT
|
8.2 | IC50 | 5 | — | |
AZCFROYDWGJIHI
|
8.2 | IC50 | 3 | — | |
HVFFRODVHZGRAZ
|
8.2 | IC50 | 4 | — | |
LIGPIGAGCDCBGQ
|
8.2 | IC50 | 2 | — | |
NRTSFXVZIHRSAM
|
8.2 | IC50 | 2 | — | |
AHCZNZBUHSRPCU
|
8.2 | IC50 | 2 | — | |
IPQLFXYRKFCCRJ
|
8.2 | IC50 | 2 | — | |
LGZFUXSDGGGPHG
|
8.2 | IC50 | 2 | — | |
WMKFJDQPAVKQAQ
|
8.1 | IC50 | 3 | — | |
LMLIBNUOIWAJFC
|
8.0 | Kd | 9 | — | |
OWQNTPSDYOZXJM
|
8.0 | IC50 | 2 | — | |
WZSQCCTZFYLIKW
|
8.0 | IC50 | 2 | — | |
ICIIHYCMSRJMHI
|
8.0 | IC50 | 2 | — | |
MYIGQQDEMVIHBG
|
7.9 | IC50 | 2 | — | |
OFWWWKWUCDUISA
|
7.9 | IC50 | 3 | — | |
MQQWUSICUOGGBD
|
7.8 | IC50 | 2 | — | |
CHEXYSJBKQQXIF
|
7.8 | IC50 | 2 | — | |
GGJRFYLWAXMCNR
|
7.8 | IC50 | 2 | — | |
CBGFEMSXMIJQKG
|
7.8 | IC50 | 3 | — | |
MOSXHKAISRXEST
|
7.8 | IC50 | 2 | — | |
PGRPAJVQVRBFEA
|
7.8 | IC50 | 2 | — | |
QAORWPLEPWLSPU
|
7.8 | IC50 | 2 | — | |
STGWRPISYALDEU
|
7.8 | IC50 | 2 | — | |
XHAYAQCABOVSNX
|
7.8 | Kd | 9 | — | |
IFILOJYOQZJYIC
|
7.8 | IC50 | 2 | — | |
UYBRROMMFMPJAN
|
7.8 | Kd | 8 | — | |
ZJQVEQKLMMZDON
|
7.8 | IC50 | 2 | — | |
LLHGUSJJGJYSJO
|
7.7 | IC50 | 2 | — | |
KZNDNGJCFUTVMP
|
7.7 | IC50 | 2 | — | |
SMABWKWHQKFGDR
|
7.6 | IC50 | 2 | — | |
UCCATIJMEOLTEL
|
7.6 | IC50 | 2 | — | |
DGXDBZHHWWZNMQ
|
7.6 | IC50 | 3 | — | |
RLNJZBANHSVNDS
|
7.5 | IC50 | 2 | — | |
VZKANYDYIVJBAM
|
7.5 | IC50 | 2 | — | |
WQPQQRVHJTZSFA
|
7.5 | IC50 | 2 | — | |
ZIQDIXVWQPULTM
|
7.5 | IC50 | 2 | — | |
IPJBCIJCPIYZEC
|
7.5 | IC50 | 2 | — | |
XQHRNYHJMOIHEB
|
7.5 | IC50 | 3 | — | |
GCGCXCUBNSDITO
|
7.4 | IC50 | 2 | — | |
XJRUWGFZGQNPPD
|
7.4 | IC50 | 3 | — | |
VNCNIMOILJQAGJ
|
7.3 | IC50 | 2 | — | |
WEIQLZUSEUMRIG
|
7.3 | IC50 | 2 | — | |
BTTCKSLDCMBUAH
|
7.3 | Ki | 7 | — | |
NDEORODKVUYMFQ
|
7.3 | Kd | 9 | — |