Target Details
| UniProt AC | P21453 |
|---|---|
| Gene Symbol | S1PR1 |
| Protein Name | Sphingosine 1-phosphate receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (4)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PMGFMZNAXWTMIY
|
6.6 | IC50 | 2 | — | |
YNUQWTWRORYOFY
|
6.6 | IC50 | 2 | — | |
TXWZXPYJUFAJOH
|
6.6 | IC50 | 2 | — | |
IXKFXZZVAFLDCK
|
6.5 | IC50 | 2 | — | |
XTPRWWYDWAJRJF
|
6.5 | IC50 | 2 | — | |
GOKJFEMIQDBPSQ
|
6.5 | IC50 | 2 | — | |
KLIRFQNFFXBULP
|
6.5 | IC50 | 2 | — | |
LKCNOGUUCKOMBY
|
6.5 | IC50 | 3 | — | |
ALKGNTQLVMWJRY
|
6.5 | IC50 | 2 | — | |
IHJCKBWPCNFLBM
|
6.5 | IC50 | 5 | — | |
HYNPQYPWKPNEIV
|
6.5 | IC50 | 2 | — | |
IHJCKBWPCNFLBM
|
6.5 | IC50 | 5 | — | |
PJFAXNXMPMOEFZ
|
6.5 | IC50 | 2 | — | |
LSZRFUXALRHLHB
|
6.4 | IC50 | 3 | — | |
MVIUMKOQNNKAJB
|
6.4 | IC50 | 2 | — | |
WAAWETUDFSIYSD
|
6.4 | IC50 | 3 | — | |
IYOSQHIKGBCWAG
|
6.4 | IC50 | 2 | — | |
LDBXYKHBFJYNLA
|
6.4 | IC50 | 2 | — | |
MZUADFOUZQOZIK
|
6.4 | IC50 | 2 | — | |
RZMNWEVQRMOJTQ
|
6.4 | IC50 | 2 | — | |
WBTSGSPPSRSUTC
|
6.4 | IC50 | 2 | — | |
DSWRSIFZAROYJS
|
6.4 | IC50 | 2 | — | |
PVDWCIKCLKCZEB
|
6.4 | IC50 | 2 | — | |
XHLMGIHCPHRVLJ
|
6.4 | IC50 | 2 | — | |
ZRXGROOHYIFHII
|
6.4 | IC50 | 2 | — | |
TUGMSRZTHAPOKQ
|
6.4 | IC50 | 2 | — | |
DIKZDUVGAXUODC
|
6.3 | IC50 | 2 | — | |
IWEBRWJRUHNDER
|
6.3 | IC50 | 2 | — | |
RTRRFXYPPMHFLR
|
6.3 | IC50 | 2 | — | |
ZQUQFQGNDHGASO
|
6.3 | IC50 | 2 | — | |
XXMKBPNOZNEJIM
|
6.3 | IC50 | 2 | — | |
BTPFDZGBSFFCLT
|
6.3 | IC50 | 2 | — | |
MOMSMTBACXQOPD
|
6.3 | IC50 | 2 | — | |
ZNZSUFLUKZCULU
|
6.3 | IC50 | 2 | — | |
FCKYVAHKARMLCH
|
6.3 | IC50 | 2 | — | |
RHJHXSBYHQEFDQ
|
6.3 | IC50 | 2 | — | |
AZUXUQTVQJSFCZ
|
6.2 | IC50 | 2 | — | |
XTEYPDFMLGCQTR
|
6.2 | IC50 | 2 | — | |
QFOCANKLYFGGDQ
|
6.2 | IC50 | 2 | — | |
QQBGLNPPVXQYJV
|
6.2 | IC50 | 2 | — | |
ZXKVNTFFHSRCQM
|
6.2 | IC50 | 2 | — | |
YILYDYRSTBZITD
|
6.2 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
6.2 | IC50 | 3 | — | |
QCIWYUKBPSHJKD
|
6.2 | IC50 | 2 | — | |
NKQKSPQAKIHFMF
|
6.2 | IC50 | 2 | — | |
UUODWPRHRNIITI
|
6.2 | IC50 | 2 | — | |
XIJOBJBWOPBBNG
|
6.1 | IC50 | 3 | — | |
GRHKCGSXHAHSFS
|
6.1 | IC50 | 2 | — | |
BJGWGOSQTOUYFH
|
6.1 | IC50 | 2 | — | |
KLZLCOULUPUMAI
|
6.1 | IC50 | 3 | — |