Target Details
| UniProt AC | P21453 |
|---|---|
| Gene Symbol | S1PR1 |
| Protein Name | Sphingosine 1-phosphate receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (4)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RMVXQVRSCUGPMJ
|
7.3 | IC50 | 2 | — | |
SUDIYZHHZHUABB
|
7.3 | IC50 | 2 | — | |
TZEMKQKSWRONQO
|
7.3 | IC50 | 2 | — | |
UAIOHVGTNPZFOZ
|
7.3 | IC50 | 2 | — | |
UESBQQDTMRKMNH
|
7.3 | IC50 | 2 | — | |
UKZOBTBQDYEIJI
|
7.3 | IC50 | 2 | — | |
UKZOBTBQDYEIJI
|
7.3 | IC50 | 2 | — | |
UMGWWSCTACWGIW
|
7.3 | IC50 | 2 | — | |
VEBJRUVXHMIZLY
|
7.3 | IC50 | 2 | — | |
VFIMMQWDLUMYOS
|
7.3 | IC50 | 2 | — | |
WHNXCKWIIZRITG
|
7.3 | IC50 | 2 | — | |
XBPWSCOKZCXAOD
|
7.3 | IC50 | 2 | — | |
XSCSVCWQFKDITI
|
7.3 | IC50 | 2 | — | |
XVMRSJJSMMSLRC
|
7.3 | IC50 | 2 | — | |
YMFWUPKLBPDNRH
|
7.3 | IC50 | 2 | — | |
CDZQINDPHHFTHS
|
7.2 | IC50 | 2 | — | |
XXVGJGHFHPWZAV
|
7.1 | IC50 | 2 | — | |
GFAWKWDBAGVYFO
|
7.1 | IC50 | 4 | — | |
IHLGWTMHFNRKTD
|
7.1 | IC50 | 3 | — | |
HBDKLCRIRSOTTL
|
7.1 | IC50 | 2 | — | |
QJQFJIOSLMKJMG
|
7.0 | IC50 | 4 | — | |
CCKXTEGCXIXMQR
|
7.0 | IC50 | 2 | — | |
MSESTOOFLKUAQK
|
7.0 | IC50 | 2 | — | |
BNVXTRHZRYNIIM
|
7.0 | IC50 | 2 | — | |
WBMGSDGYARVKJE
|
7.0 | IC50 | 2 | — | |
KOMZDIJMFFDGRK
|
6.9 | IC50 | 2 | — | |
VHKORLDZIRFKDI
|
6.9 | IC50 | 2 | — | |
DTNQUUSARXMSRT
|
6.9 | IC50 | 2 | — | |
JWFPFBZCDCVFBO
|
6.8 | IC50 | 2 | — | |
GRBYKZJOZJYFPB
|
6.8 | IC50 | 3 | — | |
LXEVGUDWNJFVRH
|
6.8 | IC50 | 2 | — | |
KKOSHWJEFBAPQK
|
6.8 | IC50 | 4 | — | |
XNKYXYWPDUHBSC
|
6.8 | IC50 | 3 | — | |
NKVZUMRBOPLFQI
|
6.8 | IC50 | 2 | — | |
CDZQINDPHHFTHS
|
6.7 | IC50 | 2 | — | |
BPFTXGAARBAJDP
|
6.7 | IC50 | 4 | — | |
LITUICLXUCBGQY
|
6.7 | IC50 | 2 | — | |
KOLOJHLHPQFMTO
|
6.7 | IC50 | 2 | — | |
QOYPZFURCHEYHM
|
6.7 | IC50 | 2 | — | |
UBEBIMAOSJLCDX
|
6.7 | IC50 | 3 | — | |
XOLPRYJQLCWVOK
|
6.7 | IC50 | 2 | — | |
QEQDYKXCRPIRTN
|
6.7 | IC50 | 2 | — | |
BBSVRUBPFGPMDU
|
6.7 | IC50 | 2 | — | |
DCJHQXHJMFDIMV
|
6.7 | IC50 | 2 | — | |
FXUWQRWIQRYKKB
|
6.7 | IC50 | 3 | — | |
IUOXTZXENSYXDS
|
6.7 | IC50 | 2 | — | |
VETBKPDTHQZBKH
|
6.7 | IC50 | 3 | — | |
QDBJDRNNPPZVNE
|
6.6 | IC50 | 2 | — | |
FODHWOBAQBTTFS
|
6.6 | IC50 | 6 | — | |
DBFCGNXJRISFMI
|
6.6 | IC50 | 4 | — |