Target Details
| UniProt AC | P21453 |
|---|---|
| Gene Symbol | S1PR1 |
| Protein Name | Sphingosine 1-phosphate receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (4)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XXVGJGHFHPWZAV
|
7.8 | IC50 | 3 | — | |
PLUJPPMSHJDKIV
|
7.8 | IC50 | 2 | — | |
GIEZYZUMOZGBGB
|
7.7 | IC50 | 2 | — | |
OVHZTRSKNATTNM
|
7.7 | IC50 | 2 | — | |
XPZPTGRFTGBSAI
|
7.7 | IC50 | 4 | — | |
JXGNTXCFTVWCAS
|
7.7 | IC50 | 2 | — | |
WMLSDMINRWPYKX
|
7.7 | IC50 | 3 | — | |
CSMQUILOGPIVIK
|
7.6 | IC50 | 2 | — | |
DHVYHNBDKXSJGJ
|
7.6 | IC50 | 2 | — | |
XZWUWZDFEBVUJQ
|
7.6 | IC50 | 4 | — | |
VRAGHPQXFBYHBQ
|
7.5 | IC50 | 2 | — | |
ATXJVJPQVHFGIA
|
7.5 | IC50 | 4 | — | |
CQHLHKGLJUEABQ
|
7.5 | IC50 | 2 | — | |
FMLHSOGKNHADEE
|
7.5 | Ki | 2 | — | |
MYSPJHRAIVKWQS
|
7.5 | Ki | 2 | — | |
ZJVUUEPNFHMZKC
|
7.5 | IC50 | 2 | — | |
AMJOZICHTKJDOI
|
7.5 | IC50 | 3 | — | |
CRSDAUWBRRWRFZ
|
7.5 | IC50 | 2 | — | |
RFNNVHCCTIWJLY
|
7.4 | IC50 | 4 | — | |
GJSCDTCSBXBNCQ
|
7.4 | IC50 | 3 | — | |
HBOVZSYNTFEZBX
|
7.3 | IC50 | 2 | — | |
LXEVGUDWNJFVRH
|
7.3 | IC50 | 2 | — | |
VYEUIGPXJOJLRN
|
7.3 | IC50 | 4 | — | |
ZEIHEVGZGIEZLO
|
7.3 | IC50 | 4 | — | |
ZUZDTPVPNQRGSJ
|
7.3 | IC50 | 4 | — | |
AEIHCANYZUEHOR
|
7.3 | IC50 | 2 | — | |
CBORBAPYEZAXSL
|
7.3 | IC50 | 2 | — | |
DDYCHYOORUTETD
|
7.3 | IC50 | 2 | — | |
DKGGXDBRTJXHDG
|
7.3 | IC50 | 2 | — | |
DMKJHQYXMABWKG
|
7.3 | IC50 | 2 | — | |
DOTOOAWYGBKVSM
|
7.3 | IC50 | 2 | — | |
DOTOOAWYGBKVSM
|
7.3 | IC50 | 2 | — | |
FDVYOQMHWPIULW
|
7.3 | IC50 | 2 | — | |
HBBFAKPITZTLRX
|
7.3 | IC50 | 2 | — | |
HPFZRSRAOKLYSR
|
7.3 | IC50 | 2 | — | |
JZNRDZRTKICFGB
|
7.3 | IC50 | 2 | — | |
KNEVIKYHXJJRPI
|
7.3 | IC50 | 2 | — | |
KRPLSASCBICFGK
|
7.3 | IC50 | 2 | — | |
KUAZUCUOHDSDFG
|
7.3 | IC50 | 2 | — | |
KUGVAWOYKCMQNB
|
7.3 | IC50 | 2 | — | |
KWRRNBCZIGUXKL
|
7.3 | IC50 | 2 | — | |
LMYHLCLZWOIUDH
|
7.3 | IC50 | 2 | — | |
MJKUOBXNYRXRCS
|
7.3 | IC50 | 2 | — | |
MJKUOBXNYRXRCS
|
7.3 | IC50 | 2 | — | |
MRWIFBGTMSTWMC
|
7.3 | IC50 | 2 | — | |
NZKZHORILZMUBN
|
7.3 | IC50 | 2 | — | |
OMCDALGIBJYJLI
|
7.3 | IC50 | 2 | — | |
OMCDALGIBJYJLI
|
7.3 | IC50 | 2 | — | |
ONQONXLWPSHUIY
|
7.3 | IC50 | 2 | — | |
RGGPEWLTXQYSJR
|
7.3 | IC50 | 2 | — |