Target Details
| UniProt AC | P21453 |
|---|---|
| Gene Symbol | S1PR1 |
| Protein Name | Sphingosine 1-phosphate receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (4)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LGOMWSIGEIXWPD
|
8.4 | IC50 | 3 | — | |
WGFVGWMDSCSXKT
|
8.4 | IC50 | 3 | — | |
WECRLAZSZWCWDE
|
8.4 | IC50 | 5 | — | |
KNLPKQCGTFMRRN
|
8.4 | IC50 | 2 | — | |
BPANWCJVYBGZFM
|
8.4 | IC50 | 4 | — | |
QEBXXPLHWMZIKW
|
8.3 | IC50 | 3 | — | |
TXPQNUNBAQRPEW
|
8.3 | IC50 | 2 | — | |
WUXNTVXUIHVAQN
|
8.3 | IC50 | 2 | — | |
AQMRGNZDLUYITB
|
8.3 | IC50 | 3 | — | |
JAMOPMAEOMFXHF
|
8.3 | IC50 | 4 | — | |
OPWNVYPWPMIBGP
|
8.3 | IC50 | 2 | — | |
QMNAPCZIOKPJDQ
|
8.3 | IC50 | 3 | — | |
DOAHOEVWZUKZMM
|
8.2 | IC50 | 3 | — | |
QEBXXPLHWMZIKW
|
8.2 | IC50 | 3 | — | |
LPAUOXUZGSBGDU
|
8.2 | IC50 | 2 | — | |
TWNDWWAUVXKNMU
|
8.2 | IC50 | 4 | — | |
YMBOZHBXRGFOHL
|
8.2 | IC50 | 2 | — | |
AFPYVDIMHNINIS
|
8.2 | IC50 | 4 | — | |
IOIGVVYTXMGUFG
|
8.2 | IC50 | 2 | — | |
ODKLTWJRUVYDRU
|
8.2 | IC50 | 5 | — | |
XGFCNYXSOCFJIR
|
8.2 | IC50 | 4 | — | |
YHDAWQLKEJHZMN
|
8.2 | IC50 | 4 | — | |
WFMGEMPWKRJJHM
|
8.1 | IC50 | 3 | — | |
XDSPSYJWGHPIAZ
|
8.1 | IC50 | 4 | — | |
ZEWHUZLAFGAHQV
|
8.1 | IC50 | 3 | — | |
NEAYDTITWAMODK
|
8.1 | IC50 | 2 | — | |
YWXALJUJDPVVHS
|
8.1 | IC50 | 4 | — | |
ZGGLMGHJHZWEKX
|
8.1 | IC50 | 3 | — | |
DOAHOEVWZUKZMM
|
8.1 | IC50 | 3 | — | |
SJSQQBATFXLXQC
|
8.1 | IC50 | 3 | — | |
OXYHNSKNRIYKDI
|
8.1 | IC50 | 3 | — | |
AAEVPRISMKXZKU
|
8.1 | IC50 | 2 | — | |
AAEVPRISMKXZKU
|
8.1 | IC50 | 4 | — | |
QGDUQFMYMKUVHT
|
8.1 | IC50 | 3 | — | |
RMDMQWBLROBEJO
|
8.0 | IC50 | 3 | — | |
NUEDANFMPBYCJM
|
7.9 | IC50 | 2 | — | |
WUCGGZATYNFGIA
|
7.9 | IC50 | 4 | — | |
YTTNOAFOCBYIIG
|
7.9 | IC50 | 4 | — | |
BDXDATLHTUEDJA
|
7.9 | IC50 | 2 | — | |
DQXSYKMXKITFAL
|
7.9 | IC50 | 3 | — | |
BGPIKLDZOZBUEW
|
7.8 | IC50 | 4 | — | |
BYMIMTPDQNLDHL
|
7.8 | IC50 | 3 | — | |
RNDCUJZLFBWJHF
|
7.8 | IC50 | 3 | — | |
ZQAPROQSGXAHSW
|
7.8 | IC50 | 4 | — | |
KARRQFDDSYYFAE
|
7.8 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
7.8 | IC50 | 4 | — | |
CDEPDWBJGIUHRS
|
7.8 | IC50 | 5 | — | |
GHGMOTNOPRPKKC
|
7.8 | IC50 | 3 | — | |
NOMBGCXWXBTHTO
|
7.8 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
7.8 | IC50 | 4 | — |