Target Details
| UniProt AC | P21453 |
|---|---|
| Gene Symbol | S1PR1 |
| Protein Name | Sphingosine 1-phosphate receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (4)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZYJFERBFOURDFL
|
9.0 | IC50 | 3 | — | |
KVYQKSXTMZHEPB
|
9.0 | IC50 | 4 | — | |
NOERNAQPKCFUKL
|
9.0 | IC50 | 4 | — | |
LVLCOLBUGCDLPB
|
9.0 | IC50 | 4 | — | |
DUYSYHSSBDVJSM
|
8.9 | Ki | 5 | — | |
FSCOADFARBASQU
|
8.9 | IC50 | 4 | — | |
IOBZROVFXAOQQI
|
8.9 | IC50 | 4 | — | |
NCUVDYUSQOEZTJ
|
8.9 | IC50 | 3 | — | |
YARHFBRDYSZBIN
|
8.9 | IC50 | 3 | — | |
GCTZIVJBMHYJOP
|
8.9 | IC50 | 4 | — | |
KVWDBAIEXNLWNP
|
8.9 | IC50 | 3 | — | |
UOLFBZYNLRKEKZ
|
8.9 | IC50 | 2 | — | |
ZQHLJZUCUJZZRV
|
8.9 | IC50 | 4 | — | |
AEINVRKYWDZAKS
|
8.8 | IC50 | 3 | — | |
AKMFGWWEWTVUTP
|
8.8 | IC50 | 3 | — | |
DUYSYHSSBDVJSM
|
8.8 | IC50 | 6 | — | |
KUOMYSKEBPYIAO
|
8.8 | IC50 | 4 | — | |
BDZJQGMIIWGSHK
|
8.8 | IC50 | 4 | — | |
LDWAKTDSZSERFS
|
8.8 | IC50 | 3 | — | |
PRUUCTGBHIGGOH
|
8.8 | IC50 | 4 | — | |
GEMQKZAVXUVYBN
|
8.8 | IC50 | 3 | — | |
ZJPSQGKCYKMKSJ
|
8.8 | IC50 | 2 | — | |
ASTHITQJQQXIDF
|
8.7 | IC50 | 2 | — | |
GTZFBQFSZBMRCX
|
8.7 | IC50 | 3 | — | |
AXAGGQQXMQHIFF
|
8.7 | IC50 | 4 | — | |
DWHWJBOQZGWGJN
|
8.7 | IC50 | 2 | — | |
GNLKZOCFPXHKNV
|
8.7 | IC50 | 2 | — | |
GYRSLHWASFQOPP
|
8.7 | IC50 | 4 | — | |
IITBTBZPEPWWLP
|
8.7 | IC50 | 3 | — | |
KRYWDAJMWJBMNZ
|
8.7 | IC50 | 4 | — | |
KYHUARFFBDLROH
|
8.7 | IC50 | 2 | — | |
BWCQGMDWAWERIV
|
8.7 | IC50 | 4 | — | |
DMOOKXPSMLPOGZ
|
8.7 | IC50 | 3 | — | |
UNTMCOZQSGVJBE
|
8.7 | IC50 | 3 | — | |
LYZKFLGVDKUPAP
|
8.6 | IC50 | 4 | — | |
POPQMXAKAVJFNJ
|
8.6 | IC50 | 4 | — | |
ROTPOJPBVJTWLI
|
8.6 | IC50 | 5 | — | |
ZJPSQGKCYKMKSJ
|
8.6 | IC50 | 2 | — | |
GBAYNJCGVHFQTM
|
8.6 | IC50 | 4 | — | |
KSAATBXYGYJAQU
|
8.6 | IC50 | 4 | — | |
LPFGMPGBYMGNTK
|
8.6 | IC50 | 4 | — | |
WJTKHEJZIPMAKN
|
8.6 | IC50 | 4 | — | |
LSXRZLMJNWYNPW
|
8.6 | IC50 | 2 | — | |
NFEFCBPHVVPEHI
|
8.6 | IC50 | 2 | — | |
QTKLDIPKJJAYHB
|
8.5 | IC50 | 3 | — | |
ZJPSQGKCYKMKSJ
|
8.5 | IC50 | 2 | — | |
AHFAXNLVTHDCEY
|
8.5 | IC50 | 2 | — | |
SJSQQBATFXLXQC
|
8.5 | IC50 | 3 | — | |
CVKVCJXTRKKPRQ
|
8.5 | IC50 | 2 | — | |
BUBRUGRTGCDHOJ
|
8.4 | IC50 | 3 | — |