Target Details
| UniProt AC | P21453 |
|---|---|
| Gene Symbol | S1PR1 |
| Protein Name | Sphingosine 1-phosphate receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 0
- Avg pChEMBL 7.77
KEGG Pathways (4)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NOMBGCXWXBTHTO
|
10.0 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
10.0 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
10.0 | IC50 | 4 | — | |
GHQKYJKUIMNJCW
|
9.8 | IC50 | 4 | — | |
HMJKTOOFFPXTGY
|
9.8 | IC50 | 4 | — | |
IILANYBHYYNGJK
|
9.8 | IC50 | 5 | — | |
LRFKWQGGENFBFO
|
9.8 | IC50 | 4 | — | |
NOMBGCXWXBTHTO
|
9.8 | IC50 | 4 | — | |
PGLFYYYVMFEVNN
|
9.8 | IC50 | 4 | — | |
IYOGKTIRIRHPOH
|
9.7 | IC50 | 6 | — | |
MJFHVHNIHASYLI
|
9.7 | IC50 | 4 | — | |
WDBMBYAFMOKUJU
|
9.7 | IC50 | 4 | — | |
LXNKUNKMYYJPKD
|
9.6 | IC50 | 3 | — | |
YRLWOUXQTIDPEK
|
9.6 | IC50 | 3 | — | |
JJPKCGYTCKVOEU
|
9.6 | IC50 | 4 | — | |
KKNUGAMJKIHACQ
|
9.6 | IC50 | 4 | — | |
LCRADRCUDVEFGB
|
9.6 | IC50 | 4 | — | |
LRFKWQGGENFBFO
|
9.6 | IC50 | 5 | — | |
KLULNXUHMWEEKT
|
9.5 | IC50 | 4 | — | |
MMKMRZFTPGRQEQ
|
9.5 | IC50 | 4 | — | |
PCBMXZQDEQINJG
|
9.5 | IC50 | 4 | — | |
HXDPHSXYLHIVSE
|
9.5 | IC50 | 4 | — | |
IJFAOCYEADEWAV
|
9.5 | IC50 | 4 | — | |
PEPDHHDQCCNILN
|
9.5 | IC50 | 4 | — | |
SQBXAXYMXPCNON
|
9.4 | IC50 | 4 | — | |
WTJGTMFQALCKRT
|
9.4 | IC50 | 4 | — | |
XYFAADCQOGUWOC
|
9.4 | IC50 | 3 | — | |
YBEAJMHMAMGKBN
|
9.4 | IC50 | 3 | — | |
YIZUZSSLYPDFOC
|
9.4 | IC50 | 4 | — | |
JNAQEIPNFVZKSC
|
9.3 | IC50 | 4 | — | |
VKXANKHCILEVSX
|
9.3 | IC50 | 4 | — | |
SHQNRSGKLNMHOS
|
9.2 | IC50 | 4 | — | |
VEAJEWXYGKUGPH
|
9.2 | IC50 | 4 | — | |
QDDQIPUKAXBMBX
|
9.2 | Ki | 3 | — | |
LTSLZRLZTPLAGI
|
9.2 | IC50 | 3 | — | |
YFWUAIPFVJAYCH
|
9.2 | IC50 | 4 | — | |
RNDGTSGYNDTFOA
|
9.1 | IC50 | 4 | — | |
JBPVYJJIRRUCJU
|
9.1 | IC50 | 4 | — | |
LRFKWQGGENFBFO
|
9.1 | IC50 | 5 | — | |
WLWWQFLRNKBLQM
|
9.1 | IC50 | 2 | — | |
BLLBAGSMDDITHA
|
9.1 | IC50 | 4 | — | |
CUPKVALESCTXBT
|
9.1 | IC50 | 2 | — | |
QIPIWIXFCSCVEI
|
9.1 | IC50 | 3 | — | |
YARHFBRDYSZBIN
|
9.1 | IC50 | 3 | — | |
PZYBHVNEGCWQOZ
|
9.1 | IC50 | 2 | — | |
GTROXDSLWCVOIS
|
9.1 | IC50 | 4 | — | |
NSEVTFLGGHULPD
|
9.1 | IC50 | 4 | — | |
QIPIWIXFCSCVEI
|
9.1 | IC50 | 3 | — | |
SHISURVONRMBAW
|
9.1 | IC50 | 4 | — | |
TXFZSDIRXYGOOU
|
9.1 | IC50 | 4 | — |