Target Details
UniProt ACP21452
Gene SymbolTACR2
Protein NameSubstance-K receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 400
  • Clinical molecules 3
  • Avg pChEMBL 7.72
Top Co-occurrence Targets
Active Molecules (400)
InChIKey pChEMBL Type Targets Clinical
MQNYRKWJSMQECI 6.6 Ki 2
MQNYRKWJSMQECI 6.6 Ki 2
XIUWYQPZUOTMGU 6.5 Ki 2
ATMHFQDWDFHUDF 6.5 IC50 2
SQRIUKXVALYAKA 6.5 Ki 2
RVDBXUCLTPUWIX 6.5 Ki 2
AVEVJMZJJJDOCI 6.5 Ki 7
DDBBEPOXFYJCCQ 6.5 Ki 2
DUJCBRGUNYAAHY 6.5 Ki 2
IFPPRPWFEFODEU 6.5 Ki 2
ODPRNYGWGVRXIG 6.5 IC50 3
JRQLUGQQZPCLHN 6.5 Ki 2
JBKANADLNPFWIK 6.4 Ki 2
PDGGHHMVDHHHGY 6.4 Ki 2
NCJWLSWXMPGOIS 6.4 IC50 3
KYEAUAKSYSOFSP 6.4 Ki 2
ORMFBQJKAWHTKC 6.4 Ki 2
ARGUIKFIPCGABR 6.4 Ki 2
BEWCDVTWUFJSSM 6.4 Ki 2
BHCJHYIMNHXLOM 6.3 Ki 2
GYVLRBXEOLZDJP 6.3 Ki 2
CTETYYAZBPJBHE 6.3 Ki 11
FBKJXYVRFOSKLQ 6.3 IC50 2
JMEKLKBPAWJBOV 6.3 Ki 3
DHUATBAZHILHIC 6.3 IC50 5
ZDZOTLJHXYCWBA 6.3 Ki 19
GBABOYUKABKIAF 6.3 Ki 17
PGOKBMWPBDRDGN 6.3 Ki 8
WBKRXYVTNUALQH 6.3 IC50 2
YQHKVGJQICUJMY 6.3 IC50 2
KLFRSZNXCXNAGN 6.2 Ki 2
UJOSAVYAWJYRDR 6.2 IC50 2
ZVBLMUFWEBYUFD 6.2 IC50 2
HLBLLGYOMVQROQ 6.2 Ki 2
USCBMUJHCSEWHX 6.2 Kd 2
MJJALKDDGIKVBE 6.2 Ki 30 Yes
SIYLLGKDQZGJHK 6.2 Ki 13
HXKFHHNEFCZKPG 6.2 IC50 3
XXUOOQREUFQRJA 6.1 IC50 2
XXUOOQREUFQRJA 6.1 IC50 2
SVJLECBANPOFKI 6.1 Ki 2
ZSIQAOCNFRWDNJ 6.1 Ki 2
NCDNCNXCDXHOMX 6.1 Ki 12
GUGOEEXESWIERI 6.0 Ki 18 Yes
NWNXAOPJFFMSJS 6.0 IC50 2
OZJDKUMSRQSURZ 6.0 Ki 3
BZWOCMMJHXYQGW 6.0 Ki 2
GXDALQBWZGODGZ 6.0 Ki 21 Yes
HMXDWDSNPRNUKI 6.0 Ki 72
PFOMIAQBONXLRP 6.0 IC50 2
2D structure