Target Details
UniProt ACP21452
Gene SymbolTACR2
Protein NameSubstance-K receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 400
  • Clinical molecules 3
  • Avg pChEMBL 7.72
Top Co-occurrence Targets
Active Molecules (400)
InChIKey pChEMBL Type Targets Clinical
YYLWLQSLLOQPBL 8.5 Ki 2
VWROPOCOVOHGMQ 8.5 Ki 2
XTUKHLMHDAVVDE 8.4 Ki 3
GLFJJJVLKJNYOY 8.4 IC50 2
FZNRYDBDVZSZBQ 8.4 Ki 2
LCMYTAQFJIXBCQ 8.4 IC50 2
MTGCTWAUNJMIJB 8.4 Ki 2
NFVAMSHCYQJREM 8.4 Ki 3
RMPKGCQPPWICCB 8.4 Ki 2
SNDJRJPQSWPPJP 8.4 Ki 2
AXBSORLKLUGMEI 8.4 Ki 3
BYIHDKGDBKWQLV 8.4 Ki 2
DJKJVWJQAVGLHJ 8.4 IC50 8
KULZXADAJUBWTD 8.4 Ki 2
MQCWKTYZKLSDJX 8.3 Ki 2
KQCIBGUILOITBS 8.3 Ki 3
DHWCQNWUMKKLBS 8.3 Ki 2
LZETVSMMDKRIBU 8.3 Ki 3
MUQJKGMXKAWCJF 8.3 Ki 2
NXAMGJRLSKEHIL 8.3 Ki 3
FELFRZJBPKZKAO 8.3 Ki 2
DMPBNZKYHOVYRU 8.3 Ki 3
AOHIJPJMMHXDHP 8.3 Ki 2
BHCJHYIMNHXLOM 8.3 IC50 2
KKLMRJSMWOEEFA 8.3 IC50 2
IUHUKZRXWQPIFE 8.2 Ki 3
JFCGXHNAIMSZNV 8.2 Ki 2
NAUMGBBZLWYADU 8.2 Ki 2
RNLBAKIMAUIWHO 8.2 Ki 2
KGORHDRKRVOPJF 8.2 Ki 2
ADXFJIYJEFFOSY 8.2 IC50 3
IILGQXXXFXWYDL 8.2 Ki 2
CDLIUHVXEYVLGX 8.2 IC50 2
CAHGELRDKXVTKA 8.2 IC50 2
JMIKNHGMALLEMU 8.2 IC50 2
ORMFBQJKAWHTKC 8.2 Ki 2
OYKIXMQKLMUJEK 8.2 IC50 3
QBBGNPIZYIFEFU 8.2 Ki 2
QMQONIJKFSQSNN 8.2 Ki 2
XNVWNVRFENUWFF 8.2 Ki 2
ZDJFLHCNTGAWQS 8.2 IC50 2
JSYXGDWNKVWMQZ 8.1 Ki 2
QAIJDUKQZAHNMO 8.1 Ki 2
SUIAZXTYRYLIFJ 8.1 Ki 2
WSYQSMJFBSIBRN 8.1 Ki 2
WZMVQZJKOVPVGZ 8.1 IC50 2
WZMVQZJKOVPVGZ 8.1 IC50 4
IKHGNAJUVAULNG 8.1 Ki 2
SGBDUEZXJHDZIY 8.1 Ki 2
BQVBUTSGRMTRRM 8.1 Ki 2
2D structure