Target Details
UniProt ACP21452
Gene SymbolTACR2
Protein NameSubstance-K receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 400
  • Clinical molecules 3
  • Avg pChEMBL 7.72
Top Co-occurrence Targets
Active Molecules (400)
InChIKey pChEMBL Type Targets Clinical
RPTJPWCOBZLMMD 9.0 IC50 3
HNYCTUJIKKNHPR 8.9 Ki 3
KYIGOCCCBXRHNJ 8.9 IC50 43
LMJTUYSCJIQXFP 8.9 Ki 3
OFUFYXNPWNFQBY 8.9 Ki 3
VMUJISIYYNPJBE 8.9 Ki 3
VVQLVPFUZGSGAS 8.9 Ki 2
HOLYVOXJFVZCRT 8.9 Ki 2
KIZBDFRCUJNMND 8.9 Ki 2
XRDBPVZKKASWBW 8.8 Ki 2
HEAUFJZALFKPBA 8.8 IC50 3
CTPXPFZFOWJXMU 8.8 Ki 2
QBQWUWIDZFTTLW 8.8 Ki 3
SDCLQZSZNIDDCP 8.8 Ki 3
BIMJVPXBEXJSPH 8.8 Ki 3
CXFWIZDXIZCABO 8.8 Ki 2
FRDDXKUSVLZWRL 8.8 Ki 3
KMXLXHFSSQDIGC 8.8 IC50 3
WEDUTVAKPIVEEC 8.8 Ki 2
PGKXDIMONUAMFR 8.8 Ki 3
AXOFNMUYIHBQIG 8.7 Ki 3
FYSFILDCEYJVBF 8.7 IC50 3
HIAJKTDCGCVKRZ 8.7 Ki 2
HPNPIPKYYHLBEB 8.7 Ki 2
LIXRIEAGLPGVJF 8.7 IC50 3
LYOBOZHSPINFAT 8.7 Ki 2
TUUDVKRGCJZJKQ 8.7 Ki 2
VUIKXPLLVYTQIQ 8.7 Ki 2
AJOJKKFFFUNGLX 8.7 IC50 2
CCRJBODRXVWELY 8.7 IC50 2
ZLPGKEGAFJLKOK 8.7 IC50 3
JMIKNHGMALLEMU 8.6 IC50 2
OAVNGCZBHRXUGH 8.6 IC50 3
FLNYCRJBCNNHRH 8.6 Ki 3
GNFGMQJCVYXXRO 8.6 IC50 2
SUCQKPUTZDUCKO 8.6 Ki 3
HSRXPFPQSJNQHE 8.6 Ki 3
KKNABYYXFGGHEP 8.6 Ki 3
VIGYJJFBPARTJM 8.6 IC50 3
UNTOMAYRJHGHHU 8.6 Ki 3
AEJFLHAKYANRRV 8.6 Ki 2
RQVBYRWUISROIZ 8.6 Ki 3
FXNGKZKTNZFAQF 8.5 Ki 2
KPOSFDMDKKTTBT 8.5 Ki 2
WFWJOZNEVLNHAC 8.5 Ki 2
QQEUFCBFNCEBTH 8.5 Ki 3
XFZQPQNPSOTOAL 8.5 Ki 2
NOGCECXKCJDXDN 8.5 Ki 2
VNPVPFKEORALML 8.5 Ki 2
MUQJKGMXKAWCJF 8.5 Ki 2
2D structure