Target Details
UniProt ACP21452
Gene SymbolTACR2
Protein NameSubstance-K receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 400
  • Clinical molecules 3
  • Avg pChEMBL 7.72
Top Co-occurrence Targets
Active Molecules (400)
InChIKey pChEMBL Type Targets Clinical
BZFUZGJXYGIQSB 10.0 Ki 2
FKXMTDOSYPOSDS 9.8 Ki 2
UZIMPODCTDOSBR 9.7 Ki 3
JCJPMSLGXSUYHY 9.7 IC50 2
WYMUYTPWSDFTKB 9.7 IC50 2
YGWRUECJIONJNP 9.7 IC50 2
LQRMREXDSWNGEJ 9.6 IC50 2
NAEMOVQWYAJZGQ 9.6 IC50 2
UUPZBGPDEPZRNL 9.6 IC50 2
RPTJPWCOBZLMMD 9.5 IC50 2
VHQVJYKYAGBACO 9.5 Ki 3
GVVCESGMKYLPQX 9.4 Ki 3
IWAUTRZUTAWFDX 9.4 Ki 3
UITMLIVWRRGLLR 9.4 Ki 3
UITMLIVWRRGLLR 9.4 Ki 3
VVRNZKKUOWFMOX 9.3 IC50 3
PGKXDIMONUAMFR 9.3 IC50 2
JHELCNUBUCOOEC 9.3 Ki 3
OPGIRYHKVMNCBN 9.3 Ki 3
ROETYKQAPNITRN 9.3 Ki 3
SARPBFWIJDNMRR 9.3 Ki 2
OAVNGCZBHRXUGH 9.2 IC50 2
PDGYBCXJKZHOPO 9.2 Ki 2
CFDNUNSOUUFTQO 9.2 Ki 2
SJHZTGDJTIZMSK 9.2 Ki 3
HEAUFJZALFKPBA 9.2 Ki 3
AXFMOMFMMVHXGZ 9.2 Ki 3
CWMJXUYOMKBSDT 9.2 Ki 3
FRVGAQVTZNXIME 9.2 Ki 3
SARPBFWIJDNMRR 9.2 Ki 2
XUGHCVWAIHDURA 9.2 Ki 3
GUIGWNGIQKNZBN 9.1 IC50 2
HLSABUHKBONAJY 9.1 Ki 2
IHIXHRXOBUMHTB 9.1 Ki 2
NBJOVNZRQQUMDG 9.1 Ki 3
NJYXPRQYHXQQOR 9.1 Ki 2
PLMUPHYPECRQJW 9.1 IC50 3
WBTKINCCINTBEY 9.1 Ki 3
ZOWPPIOEPFAGCI 9.1 Ki 3
WQUXLRVVRRBKCO 9.1 IC50 2
CGWJCDGSTFDBEP 9.1 Ki 3
KSZGGGOZKNJLSY 9.1 Ki 3
PTIYKSDBVLRZAO 9.1 Ki 2
RTUNBOPBBCULLC 9.0 Ki 2
UFOHFERURWEZAP 9.0 Ki 2
WAKWRTKDSYUGIM 9.0 Ki 2
ZZFJEAWXKJAJIS 9.0 Ki 3
AKWFEANKAWGNIH 9.0 Ki 2
BEMWOCKAHZVMIH 9.0 Ki 3
NOGCECXKCJDXDN 9.0 Ki 2
2D structure