Target Details
| UniProt AC | P20831 |
|---|---|
| Gene Symbol | gyrA |
| Protein Name | DNA gyrase subunit A |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 207
- Clinical molecules 0
- Avg pChEMBL 7.25
Active Molecules (207)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IDBNSMFFTLKKMN
|
6.8 | IC50 | 4 | — | |
PZFAZQUREQIODZ
|
6.8 | IC50 | 2 | — | |
ACCKRUPDYNOTMI
|
6.7 | IC50 | 2 | — | |
NHXTWWVJRWMAAW
|
6.7 | IC50 | 4 | — | |
GOMYQMSOGFDKOC
|
6.7 | IC50 | 2 | — | |
PTUWCOMLTLLKMO
|
6.7 | IC50 | 2 | — | |
USGHRRVFKSLEJT
|
6.7 | IC50 | 4 | — | |
BCOYDHFZZXSZFA
|
6.7 | IC50 | 3 | — | |
JRAGTUWUNIDVFX
|
6.7 | IC50 | 4 | — | |
QUTCIOKBWBLIHI
|
6.7 | IC50 | 2 | — | |
VINPUJZJRCEBET
|
6.7 | IC50 | 5 | — | |
FGJQMRKSDIRTPZ
|
6.6 | IC50 | 2 | — | |
KDGQBAIMBSYHIS
|
6.6 | IC50 | 4 | — | |
CYZXIGIUUJGEAZ
|
6.6 | IC50 | 2 | — | |
OKENRSAOABWGQG
|
6.6 | IC50 | 2 | — | |
HPAZHEGIKZGDCM
|
6.6 | IC50 | 2 | — | |
JCIZDZAGSUATFA
|
6.6 | IC50 | 2 | — | |
QUDWUIDMIRCCRB
|
6.6 | IC50 | 4 | — | |
CHZUNXJHDDAQCN
|
6.5 | IC50 | 2 | — | |
GGBBBGOHXWJLMT
|
6.5 | IC50 | 2 | — | |
XSSZBMPRNHMAKY
|
6.5 | IC50 | 2 | — | |
YOYJNWLSAZAWII
|
6.5 | IC50 | 2 | — | |
MTXGSGLDYXIXFF
|
6.5 | IC50 | 2 | — | |
NJYBFGSBBSLYJT
|
6.5 | IC50 | 2 | — | |
FBPOTAKJJMHABF
|
6.5 | IC50 | 2 | — | |
XSXONJWDSRZBAF
|
6.5 | IC50 | 2 | — | |
NIYHGMQLZAKUHX
|
6.4 | IC50 | 2 | — | |
WAEUAYAUPYCHGQ
|
6.4 | IC50 | 2 | — | |
FMRGAIDONMILDD
|
6.4 | IC50 | 2 | — | |
LSJGLPVZTDCYHQ
|
6.4 | IC50 | 2 | — | |
NAIYBWHMNBAOOG
|
6.4 | IC50 | 2 | — | |
PVQZLFGKXHAYPL
|
6.4 | IC50 | 2 | — | |
ZPMXCTSMZFCELU
|
6.4 | IC50 | 2 | — | |
LTAIYJYCNFSYJU
|
6.4 | IC50 | 2 | — | |
SHKVDXCLBNOXFB
|
6.3 | IC50 | 4 | — | |
FWSHCMNGNALZOS
|
6.3 | IC50 | 2 | — | |
NVTFDVCDEYDKOF
|
6.3 | IC50 | 2 | — | |
BUTXZCVRZRLABV
|
6.3 | IC50 | 2 | — | |
DSDOZOZJMRNMPG
|
6.3 | IC50 | 2 | — | |
GUEBWQFTJDQZMH
|
6.3 | IC50 | 2 | — | |
LRWFDEKCPDECFN
|
6.3 | IC50 | 2 | — | |
BIXHRRHYTOOQAX
|
6.3 | IC50 | 2 | — | |
VNAUIRAHNMVVSZ
|
6.3 | IC50 | 2 | — | |
IKVHDDZQOIVFJG
|
6.2 | IC50 | 2 | — | |
GIWUNNJISQFQLW
|
6.2 | IC50 | 2 | — | |
ZCCQPOJAEYPDRY
|
6.2 | IC50 | 2 | — | |
ILSQZDCVJPCWKM
|
6.2 | IC50 | 2 | — | |
LYHIOGOWOBGMBW
|
6.2 | IC50 | 2 | — | |
ZUZQMIMKRITPON
|
6.2 | IC50 | 2 | — | |
CECJUHKZSOSOJJ
|
6.2 | IC50 | 2 | — |