Target Details
| UniProt AC | P20831 |
|---|---|
| Gene Symbol | gyrA |
| Protein Name | DNA gyrase subunit A |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 207
- Clinical molecules 0
- Avg pChEMBL 7.25
Active Molecules (207)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MCUJWFPIOPLDLN
|
7.2 | IC50 | 2 | — | |
UYUKGVMPADBCHE
|
7.2 | IC50 | 2 | — | |
YERDVHADHPXHFF
|
7.2 | IC50 | 4 | — | |
ZFMCWMJGTDHLKI
|
7.2 | IC50 | 2 | — | |
ZFMCWMJGTDHLKI
|
7.2 | IC50 | 4 | — | |
SEAMOYQPPFJZJR
|
7.2 | IC50 | 2 | — | |
VSRUEFVCYYXLCL
|
7.2 | IC50 | 4 | — | |
KLRROQBNYDDGAK
|
7.2 | IC50 | 2 | — | |
NNEBZSDVZCUBGK
|
7.2 | IC50 | 2 | — | |
OWUGLCKBNARAPP
|
7.2 | IC50 | 2 | — | |
OTZGDJFOSDFRBQ
|
7.1 | Ki | 2 | — | |
LHPGCGRDVFMGGQ
|
7.1 | IC50 | 2 | — | |
JHJANKDCEYKCQY
|
7.0 | IC50 | 4 | — | |
LMBMQPCDCXNUGI
|
7.0 | IC50 | 2 | — | |
PNXMNHGKWCLCMU
|
7.0 | IC50 | 4 | — | |
WMNKVDSSYPIFBR
|
7.0 | IC50 | 2 | — | |
PQWWHNZAZANFOZ
|
7.0 | IC50 | 5 | — | |
CZTMTIJJNWLREO
|
7.0 | IC50 | 2 | — | |
RSJIYODUVAGVDD
|
7.0 | IC50 | 2 | — | |
MCMNYTOHUPZLOA
|
6.9 | IC50 | 5 | — | |
IYDSEXALBFJDID
|
6.9 | IC50 | 2 | — | |
BMANDSXMIVZGEY
|
6.9 | IC50 | 2 | — | |
KFEYIAJIUJJIRU
|
6.9 | IC50 | 2 | — | |
AUXHQPYDIVPJQT
|
6.9 | IC50 | 2 | — | |
DNYLEYUAAXOKIE
|
6.9 | IC50 | 2 | — | |
FBUOCINPAWXYMK
|
6.9 | IC50 | 2 | — | |
GUEBWQFTJDQZMH
|
6.9 | IC50 | 2 | — | |
HDUOQGPJPLEPTI
|
6.9 | IC50 | 2 | — | |
IGGQZENFMDGPEU
|
6.9 | IC50 | 2 | — | |
NDXWAAKFUDDIDP
|
6.9 | IC50 | 2 | — | |
OCZXFLPYVJPVBO
|
6.9 | IC50 | 2 | — | |
PEKRPORMYGTOHQ
|
6.9 | IC50 | 4 | — | |
ROYGGNJCSVBHRS
|
6.9 | IC50 | 2 | — | |
RXUHYHMLLDSVIR
|
6.9 | IC50 | 2 | — | |
STJYMKNNSABJJZ
|
6.9 | IC50 | 2 | — | |
STVLAIOEZXTGBZ
|
6.9 | IC50 | 2 | — | |
VQIOYVHLFZXJKX
|
6.9 | IC50 | 2 | — | |
VRARNXIVPHOALP
|
6.9 | IC50 | 2 | — | |
WCUIUMSVLSFGOF
|
6.9 | IC50 | 2 | — | |
WTWWYEPNQHNZPG
|
6.9 | IC50 | 2 | — | |
YXBBGIQQSYFFLN
|
6.9 | IC50 | 2 | — | |
RXPOVSSVBGRCOL
|
6.9 | IC50 | 2 | — | |
RXPOVSSVBGRCOL
|
6.9 | IC50 | 4 | — | |
PVXIXLXRCQEKAV
|
6.8 | IC50 | 2 | — | |
HVMVZISHQKEBLK
|
6.8 | IC50 | 4 | — | |
ASSSIFUQVIZHMH
|
6.8 | IC50 | 4 | — | |
LCOLURQRVPFTDK
|
6.8 | IC50 | 2 | — | |
MTZDGHNXQDFUTD
|
6.8 | IC50 | 2 | — | |
WPELWRSZEWXHNV
|
6.8 | IC50 | 2 | — | |
XMEXMBWRTDMDET
|
6.8 | IC50 | 2 | — |