Target Details
| UniProt AC | P20831 |
|---|---|
| Gene Symbol | gyrA |
| Protein Name | DNA gyrase subunit A |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 207
- Clinical molecules 0
- Avg pChEMBL 7.25
Active Molecules (207)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CSZPQXUAUHAYCD
|
7.8 | IC50 | 2 | — | |
IALGYKMHQTUZKU
|
7.8 | IC50 | 2 | — | |
OYMANMFQDCXOBU
|
7.7 | IC50 | 2 | — | |
NCLUNRIHYLBNFH
|
7.7 | IC50 | 2 | — | |
RPPRAYQNSDDYNW
|
7.7 | IC50 | 2 | — | |
VVEJKTJFDNJXPE
|
7.7 | IC50 | 2 | — | |
RCLQISQKEHCDJQ
|
7.7 | IC50 | 2 | — | |
ITPKAVKSJPIEAO
|
7.7 | IC50 | 2 | — | |
NHGOYZZJDWYVQI
|
7.7 | IC50 | 2 | — | |
JYWWBHCZYATUHE
|
7.6 | Ki | 3 | — | |
NOFFJHQFGONLBN
|
7.6 | IC50 | 2 | — | |
ADSSMWXJGIZKAA
|
7.6 | IC50 | 2 | — | |
KNMVXMHCKCETBH
|
7.6 | IC50 | 2 | — | |
DGQXHLCSQRKIHE
|
7.5 | IC50 | 2 | — | |
DRXUTILJOGAOMV
|
7.5 | IC50 | 2 | — | |
FHTDGAZUCMURNX
|
7.5 | IC50 | 2 | — | |
GHHOFTMHPOSKMT
|
7.5 | IC50 | 2 | — | |
GKHZEESTUIUGRF
|
7.5 | IC50 | 2 | — | |
GUEBWQFTJDQZMH
|
7.5 | IC50 | 2 | — | |
IHSQMSICYAUMDD
|
7.5 | IC50 | 2 | — | |
ITGDBTWKMCUOIO
|
7.5 | IC50 | 2 | — | |
JYJKOWWSKTWAJA
|
7.5 | IC50 | 2 | — | |
LCLDHRABJQNSRC
|
7.5 | IC50 | 2 | — | |
NBVFLYCKGZUYNY
|
7.5 | IC50 | 2 | — | |
NJRDESRTNBBMTM
|
7.5 | IC50 | 2 | — | |
QOVVLMSONAAZQW
|
7.5 | IC50 | 2 | — | |
RVRXIFHRYITMFV
|
7.5 | IC50 | 2 | — | |
TVDNDLRKUKVCCR
|
7.5 | IC50 | 4 | — | |
TWOGVSMCVZUIJI
|
7.5 | IC50 | 4 | — | |
XTVIZXPGQNSAAD
|
7.5 | IC50 | 4 | — | |
ZFHGPRXWTHXFEG
|
7.5 | IC50 | 2 | — | |
ZIEKVRDXDUZMKV
|
7.5 | IC50 | 4 | — | |
LQLWJUMWEYKNBM
|
7.5 | IC50 | 2 | — | |
IJZXBWJKPBRXAR
|
7.5 | IC50 | 4 | — | |
MLGPJPYFHAIWJL
|
7.5 | IC50 | 2 | — | |
SWRWDZXTXMXZOR
|
7.4 | IC50 | 2 | — | |
ZYUKGEKHLULSGR
|
7.4 | IC50 | 4 | — | |
WQQLMAXPGNMODY
|
7.4 | IC50 | 2 | — | |
BKRYLNPFZBMBFV
|
7.4 | IC50 | 3 | — | |
PHKHNRMHOSCRKO
|
7.4 | IC50 | 4 | — | |
YJQPYGGHQPGBLI
|
7.4 | IC50 | 2 | — | |
UHAMREUUTPXOJY
|
7.4 | IC50 | 2 | — | |
VBBHJKPBFFTRMO
|
7.4 | IC50 | 2 | — | |
NIIWFDOFEHUZBO
|
7.3 | IC50 | 4 | — | |
XQIQPWLZMBMFEZ
|
7.3 | IC50 | 2 | — | |
GFQDXSUJWFUHQT
|
7.3 | IC50 | 4 | — | |
BEOSXWIEPVUVCZ
|
7.3 | IC50 | 2 | — | |
IBUUDJJQWLQLAV
|
7.3 | IC50 | 2 | — | |
FKYJTRSZYAUQIF
|
7.2 | IC50 | 2 | — | |
HGMMQCMKBSYTFD
|
7.2 | IC50 | 2 | — |