Target Details
| UniProt AC | P20701 |
|---|---|
| Gene Symbol | ITGAL |
| Protein Name | Integrin alpha-L |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF00357 (Integrin_alpha) PF00092 (VWA) |
Summary
- Multi-target molecules 369
- Clinical molecules 0
- Avg pChEMBL 7.12
KEGG Pathways (14)
- Cell adhesion molecule (CAM) interaction
- Epstein-Barr virus infection
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Viral myocarditis
Active Molecules (369)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GMDRWNJYSVNFBO
|
6.4 | IC50 | 3 | — | |
RCJLHHUGMJBOQG
|
6.3 | IC50 | 3 | — | |
FAEVSCKIBUDMQJ
|
6.3 | IC50 | 3 | — | |
GUXYQKMGUHCFDG
|
6.3 | IC50 | 3 | — | |
XIVLZMACKMSZRH
|
6.3 | IC50 | 3 | — | |
FRTCDBYRRZDOQQ
|
6.3 | IC50 | 3 | — | |
QUFQVFKQRMTIMD
|
6.3 | IC50 | 3 | — | |
XXLJXHUHENVDCY
|
6.3 | IC50 | 3 | — | |
BYQWOSKTUPJKFV
|
6.3 | IC50 | 3 | — | |
COVPLULNDBDXTN
|
6.3 | IC50 | 3 | — | |
YZCNYQLRQDZAIE
|
6.3 | IC50 | 3 | — | |
GBOGMAARMMDZGR
|
6.3 | IC50 | 4 | — | |
JLPFLAVJCXFYQO
|
6.3 | IC50 | 3 | — | |
MTAOLVAODYGSDX
|
6.3 | IC50 | 3 | — | |
PAOXPBIXQUNYMI
|
6.3 | IC50 | 3 | — | |
KHWFLVYYKGXMPW
|
6.3 | IC50 | 3 | — | |
OLMNMKWZYAOBIK
|
6.3 | IC50 | 3 | — | |
WVTSKZKNRPBXCK
|
6.3 | IC50 | 3 | — | |
HOJGBSXDHZVYRK
|
6.2 | IC50 | 3 | — | |
GZUBGTRIHHDYOX
|
6.2 | IC50 | 3 | — | |
MOPRGMKHXDVBQR
|
6.2 | IC50 | 3 | — | |
AQVUSOQZBUOAJM
|
6.2 | IC50 | 3 | — | |
AYINYYMJNHOUSM
|
6.2 | IC50 | 3 | — | |
BDMKWKGKWYADLX
|
6.2 | IC50 | 3 | — | |
JFWCMDPBPZTELG
|
6.2 | IC50 | 3 | — | |
KEQWSKKEOZLWRV
|
6.2 | IC50 | 3 | — | |
LFNWSXGKAAHEMT
|
6.2 | IC50 | 3 | — | |
NTQOVYVRCPMWAF
|
6.2 | IC50 | 3 | — | |
SLYGCFGQHBIXPM
|
6.2 | IC50 | 3 | — | |
LXBNAFUQTGPRDK
|
6.2 | Kd | 3 | — | |
NZDSKVKNJZPPBI
|
6.2 | IC50 | 3 | — | |
PMUGSFJFKNRORH
|
6.2 | IC50 | 3 | — | |
RKPWNENDRHTTBF
|
6.2 | IC50 | 3 | — | |
YIIHVSKSGPYBER
|
6.2 | IC50 | 3 | — | |
AVYYYDWRPGSZGL
|
6.2 | IC50 | 3 | — | |
CWERXZGWAYOKSY
|
6.2 | IC50 | 3 | — | |
PUAUSJUWVGDGCP
|
6.2 | IC50 | 3 | — | |
VDCWKOMRFTYIHX
|
6.2 | IC50 | 3 | — | |
XZXXUNSFXFQLLU
|
6.2 | IC50 | 3 | — | |
JXXZCGNZJULUEM
|
6.1 | IC50 | 3 | — | |
TXMYNHMEJQOXEL
|
6.1 | IC50 | 3 | — | |
YYCCOHSORPUJOI
|
6.1 | IC50 | 3 | — | |
DEQNAOBMFIOGRH
|
6.1 | IC50 | 3 | — | |
GKARTWDJGSTNQC
|
6.1 | IC50 | 3 | — | |
MDRVMCFSALAITN
|
6.1 | IC50 | 3 | — | |
MTCSXDMZKVZCAO
|
6.1 | Kd | 3 | — | |
WBTAHXUCBNIOHJ
|
6.1 | IC50 | 3 | — | |
XYLAVJHBJRSVOB
|
6.1 | IC50 | 3 | — | |
DJXITUPRUAXMQZ
|
6.1 | IC50 | 3 | — | |
GMUWOYDXNLWCCN
|
6.1 | IC50 | 3 | — |