Target Details
| UniProt AC | P20701 |
|---|---|
| Gene Symbol | ITGAL |
| Protein Name | Integrin alpha-L |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF00357 (Integrin_alpha) PF00092 (VWA) |
Summary
- Multi-target molecules 369
- Clinical molecules 0
- Avg pChEMBL 7.12
KEGG Pathways (14)
- Cell adhesion molecule (CAM) interaction
- Epstein-Barr virus infection
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Viral myocarditis
Active Molecules (369)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZSWCQOTQDDSHT
|
8.0 | IC50 | 3 | — | |
PKSKMDBFTLPBGD
|
8.0 | IC50 | 3 | — | |
LXPIKCWBQUZGHG
|
8.0 | IC50 | 3 | — | |
OISQKZHMDXVZKJ
|
8.0 | Kd | 3 | — | |
QQSAZMAJLFVCGT
|
8.0 | IC50 | 3 | — | |
TZLWATKWJLUXTA
|
8.0 | Kd | 3 | — | |
UHTHCCFWRKLUOC
|
8.0 | IC50 | 3 | — | |
UQFJJELMTYQZLF
|
8.0 | Kd | 3 | — | |
ZFUSMHKFXKIZTH
|
8.0 | IC50 | 3 | — | |
PXWKZXMPCCTSLZ
|
8.0 | IC50 | 3 | — | |
PQEXIWGLHFOPDT
|
8.0 | IC50 | 3 | — | |
BODOXPRBLCFXNR
|
7.9 | IC50 | 3 | — | |
HCVGIQGOPCGGPD
|
7.9 | IC50 | 3 | — | |
LYDRSMBADUZQIU
|
7.9 | IC50 | 3 | — | |
LBFPLUWTLKUUCU
|
7.9 | IC50 | 3 | — | |
UNSPTWPYUISLGN
|
7.8 | IC50 | 3 | — | |
WZWKDGGJAXYHLC
|
7.8 | IC50 | 3 | — | |
XYVGXDQZIPFLPB
|
7.8 | IC50 | 3 | — | |
GKGJFUXSTSUKPB
|
7.7 | Kd | 2 | — | |
IAAIGCGTGAJLIA
|
7.7 | IC50 | 3 | — | |
WBSXKVRTVMHGNY
|
7.7 | IC50 | 3 | — | |
HXFLTJZCIRRAHJ
|
7.7 | IC50 | 3 | — | |
NPMNYUOXEKFFIQ
|
7.7 | IC50 | 3 | — | |
QIHAPYRUKBWYGW
|
7.7 | IC50 | 3 | — | |
CWQGLTCXNRXUQD
|
7.7 | Kd | 3 | — | |
FOXOPJJICTTZEU
|
7.7 | IC50 | 3 | — | |
FVEAFWBHBUVJQZ
|
7.7 | IC50 | 3 | — | |
MLYREBCRTPGARB
|
7.7 | Kd | 3 | — | |
MYIHWAVPLWUTSA
|
7.7 | Kd | 3 | — | |
SWIQOJQBTDWCRB
|
7.7 | IC50 | 3 | — | |
WVCQICGGXLHQQZ
|
7.7 | IC50 | 3 | — | |
NXNKJLOEGWSJGI
|
7.7 | IC50 | 3 | — | |
OSHCCAHIHYVBQE
|
7.7 | IC50 | 3 | — | |
FJNJHZQMQRVZEE
|
7.6 | IC50 | 3 | — | |
ZTKAYKYKKPDCAJ
|
7.6 | IC50 | 3 | — | |
AQMLUIURUPLBCR
|
7.6 | IC50 | 3 | — | |
WVKIRPXFXBGIEJ
|
7.6 | IC50 | 3 | — | |
UIQHPJBLRPBJON
|
7.6 | IC50 | 3 | — | |
QNPSGQWAWDUUBG
|
7.6 | IC50 | 3 | — | |
WHGBQVUQKROPLI
|
7.6 | IC50 | 3 | — | |
XEKXLTGSRAVVJK
|
7.6 | IC50 | 3 | — | |
JFOZKMSJYSPYLN
|
7.6 | IC50 | 3 | — | |
GWKUQIDUBUTSSN
|
7.6 | IC50 | 3 | — | |
WMECQBYXSNEKHN
|
7.6 | IC50 | 3 | — | |
CYHYOQQJILLXPV
|
7.6 | IC50 | 3 | — | |
XYTRSSKMVCVZQA
|
7.5 | IC50 | 3 | — | |
ZTROBKLFMPLYHQ
|
7.5 | IC50 | 3 | — | |
GLGFUMDYDHOFDP
|
7.5 | IC50 | 3 | — | |
IJHCQZSIRPACKX
|
7.5 | Kd | 3 | — | |
MRWGXKWDMVKCMX
|
7.5 | IC50 | 3 | — |