Target Details
| UniProt AC | P20701 |
|---|---|
| Gene Symbol | ITGAL |
| Protein Name | Integrin alpha-L |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF00357 (Integrin_alpha) PF00092 (VWA) |
Summary
- Multi-target molecules 369
- Clinical molecules 0
- Avg pChEMBL 7.12
KEGG Pathways (14)
- Cell adhesion molecule (CAM) interaction
- Epstein-Barr virus infection
- Human T-cell leukemia virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Leukocyte transendothelial migration
- Malaria
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Rheumatoid arthritis
- Staphylococcus aureus infection
- Viral myocarditis
Active Molecules (369)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VORCYKUSPCBIIJ
|
9.5 | IC50 | 3 | — | |
AXSOGTWJBSDWJQ
|
9.4 | IC50 | 3 | — | |
CAESXWPQYVXWFJ
|
9.3 | IC50 | 3 | — | |
URZCVPKXOJQTLC
|
9.3 | IC50 | 3 | — | |
AXSOGTWJBSDWJQ
|
9.2 | IC50 | 3 | — | |
SVJJYZFYKBOVBA
|
9.2 | IC50 | 3 | — | |
NVVGCQABIHSJSQ
|
9.1 | IC50 | 6 | — | |
IVAMLBGGCGJJFO
|
9.1 | IC50 | 3 | — | |
FEEFNAKFIFJCIA
|
9.0 | IC50 | 3 | — | |
RCIAZGDKPJKNPZ
|
8.9 | IC50 | 3 | — | |
BAHKPHNZYOKPQK
|
8.8 | IC50 | 3 | — | |
DMEDNZSJTBCBCR
|
8.8 | IC50 | 3 | — | |
VDABXUWSEUQIIC
|
8.8 | IC50 | 3 | — | |
KLSZVPNVFKKIRD
|
8.8 | IC50 | 3 | — | |
DZYZAGBAGWPMOE
|
8.7 | IC50 | 3 | — | |
FZYXWDXHAVNVET
|
8.7 | IC50 | 3 | — | |
VEYUKVJMTNXXSF
|
8.7 | IC50 | 3 | — | |
URZCVPKXOJQTLC
|
8.6 | IC50 | 3 | — | |
VQFPBCXPBVPOKI
|
8.6 | IC50 | 3 | — | |
ZRIKDHLPCRURPX
|
8.6 | IC50 | 3 | — | |
WBSXKVRTVMHGNY
|
8.5 | IC50 | 3 | — | |
YCCWPJKUJHZBMA
|
8.5 | IC50 | 3 | — | |
SLISYJFUVRUCKA
|
8.5 | IC50 | 3 | — | |
DMEDNZSJTBCBCR
|
8.5 | IC50 | 3 | — | |
VHJSCKJBRABOFP
|
8.5 | IC50 | 3 | — | |
VHJSCKJBRABOFP
|
8.5 | IC50 | 3 | — | |
ONDASBAVURIEBH
|
8.4 | IC50 | 3 | — | |
LLDYORSLNIEEGL
|
8.4 | IC50 | 3 | — | |
DZYZAGBAGWPMOE
|
8.4 | IC50 | 3 | — | |
BWZVEDBBEOJBAG
|
8.4 | IC50 | 3 | — | |
AIXJUFNJLMLMNA
|
8.3 | IC50 | 3 | — | |
LMKUPFOQNQUVLK
|
8.3 | IC50 | 3 | — | |
QCABIGRYALYSAQ
|
8.3 | IC50 | 3 | — | |
DMTPQLIVNVZBPV
|
8.3 | IC50 | 3 | — | |
GKORLDUEXWMZDW
|
8.2 | IC50 | 3 | — | |
MCNILTQMLDZWKD
|
8.2 | IC50 | 3 | — | |
PZFCKINMYJYVSY
|
8.2 | IC50 | 3 | — | |
WCVPXAWSKHNQTH
|
8.2 | IC50 | 3 | — | |
PEMCDDOYUUHYRN
|
8.2 | IC50 | 3 | — | |
HSJWUDLCVCZMAZ
|
8.2 | IC50 | 3 | — | |
OHELAVHWEMILBF
|
8.2 | IC50 | 3 | — | |
ZBDUGVCGVJAVEM
|
8.2 | IC50 | 3 | — | |
GYELUVCNTNLZSS
|
8.1 | IC50 | 3 | — | |
BWIPTTGMQIMVBA
|
8.1 | IC50 | 3 | — | |
SYGPJZDISKKEIV
|
8.1 | IC50 | 3 | — | |
QPWDZBBZIVDASP
|
8.1 | IC50 | 3 | — | |
XEANMEGOYUBDBY
|
8.1 | IC50 | 3 | — | |
AVUBMOWMBYBZOK
|
8.1 | Kd | 3 | — | |
MEMSOGHDJLMQDL
|
8.1 | IC50 | 3 | — | |
QOPHPRIAHZKBGU
|
8.1 | IC50 | 3 | — |