Target Details
| UniProt AC | P20366 |
|---|---|
| Gene Symbol | TAC1 |
| Protein Name | Protachykinin-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02202 (Tachykinin) |
Summary
- Multi-target molecules 13
- Clinical molecules 6
- Avg pChEMBL 6.31
KEGG Pathways (2)
Active Molecules (13)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UXSRDCKIZSWGGE
|
10.0 | Ki | 4 | — | |
AXKPFOAXAHJUAG
|
6.0 | Ki | 14 | — | |
GZKLJWGUPQBVJQ
|
6.0 | Ki | 24 | Yes | |
HDOZVRUNCMBHFH
|
6.0 | Ki | 26 | Yes | |
LNEPOXFFQSENCJ
|
6.0 | Ki | 33 | Yes | |
MVWVFYHBGMAFLY
|
6.0 | Ki | 31 | Yes | |
PMXMIIMHBWHSKN
|
6.0 | Ki | 19 | — | |
QOYHHIBFXOOADH
|
6.0 | Ki | 16 | — | |
RAPZEAPATHNIPO
|
6.0 | Ki | 28 | Yes | |
URKOMYMAXPYINW
|
6.0 | Ki | 27 | Yes | |
VSWBSWWIRNCQIJ
|
6.0 | Ki | 23 | — | |
WXPNDRBBWZMPQG
|
6.0 | Ki | 28 | — | |
ZUXABONWMNSFBN
|
6.0 | Ki | 29 | — |