Target Details
UniProt ACP20309
Gene SymbolCHRM3
Protein NameMuscarinic acetylcholine receptor M3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,440
  • Clinical molecules 32
  • Avg pChEMBL 7.8
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (1,440)
InChIKey pChEMBL Type Targets Clinical
FJVQALKRJDSNIH 9.2 IC50 3
GPSZYYQYTBZUGG 9.2 IC50 3
HIUWSDVYOJMZKY 9.2 IC50 2
IGLUHPGBUNAWCF 9.2 IC50 2
JNJKTGYSCZXDCF 9.2 IC50 3
QJBDLOQOXGQJTD 9.2 Ki 5
WRRKXJXJKFCUCR 9.2 IC50 3
QOXJSXPGWIRRNX 9.2 Ki 5
BMGXRDCNNLFFQN 9.2 Ki 2
CTFDKSWRIMHOOV 9.2 Kd 3
DKSKKVAOIPURFT 9.2 Ki 24
DVSLSPWSCJLOGG 9.2 Ki 2
GOBQSCBEINUNFL 9.2 Ki 24
GSVREIJRMHEFJP 9.2 Kd 3
HISPQXKGBMUIPU 9.2 Ki 2
LWKFTNSSJJTMGU 9.2 Ki 3
PXFIGAQEXLTGJY 9.2 Ki 2
UXEIWFVTAFVRHB 9.2 Ki 6
JXUDJJIKYUMXJI 9.2 Ki 3
YDKILWXULISVAK 9.2 Ki 2
BDWSAAGKPWOYAA 9.2 IC50 2
FYYWKHFZJYSOCA 9.2 IC50 2
NYFXIMCEKNFZKB 9.2 Ki 2
RKQTVVAARMPEBJ 9.2 Ki 2
BDWSAAGKPWOYAA 9.2 IC50 2
CBWGSRNEOFXWKO 9.2 IC50 3
CFPVEUFKLQKJRS 9.2 IC50 3
LLPYCIXHQOFZRV 9.2 IC50 3
LUSSDTRXSSFHLT 9.2 IC50 2
MKNASJNZVVEVJG 9.2 Ki 2
RBDHPXXRYPWNOU 9.2 IC50 3
KYIGOCCCBXRHNJ 9.1 IC50 43
XQODGRWXBOXGGN 9.1 IC50 3
AFLBGAQHDSOPKA 9.1 Ki 5
KXDZFZWHYIWOHI 9.1 Ki 2
DAIWBMZPSVQRCH 9.1 IC50 3
POGDAPYUQHRUOU 9.1 Ki 5
QTWQZQOULZVQSB 9.1 Ki 2
IJPOIHRHFSVJOM 9.1 Ki 3
BRWJBQIGGNWUBO 9.1 IC50 2
CFNDICOOQNMZPG 9.1 Ki 2
CXRIFSPGYWTKPW 9.1 IC50 3
FMMIDZWTNQYEIY 9.1 Ki 24
GTJTVOBMGAUNFW 9.1 Ki 2
ITYRYCDVBXJIPH 9.1 IC50 2
MVHSLDBDBCMMLB 9.1 Ki 2
PMQYZWMILDAHGO 9.1 Ki 2
RHWFCIJKMABLLH 9.1 IC50 3
RTMQZXMBCBMCJK 9.1 Ki 2
USQNTAQKHGOWIT 9.1 Ki 2
2D structure