Target Details
UniProt ACP20309
Gene SymbolCHRM3
Protein NameMuscarinic acetylcholine receptor M3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,440
  • Clinical molecules 32
  • Avg pChEMBL 7.8
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (1,440)
InChIKey pChEMBL Type Targets Clinical
RBDHPXXRYPWNOU 9.4 IC50 3
REMJCBLKEGJHMN 9.4 IC50 3
BZZXNLIQFMRDFS 9.4 Ki 2
CXURQFXHOSDLEY 9.4 Ki 2
DGTRJTZMXLDJAT 9.4 Ki 2
DUFXKHQAHBTYTO 9.4 IC50 2
KPFFPWNKWSYQFT 9.4 Ki 24
LHEDAJCFTHJHJR 9.4 Ki 2
LURMNNWUAQQCSQ 9.4 IC50 2
LVRXKANVLQJEAI 9.4 Ki 2
LVRXKANVLQJEAI 9.4 Ki 2
SXLRCJRTHFTCEE 9.4 Ki 2
VLFQTZCSVOQNQS 9.4 IC50 2
WNYTURUPCKQEMA 9.4 IC50 2
ZFSMAQQMDBOIHL 9.4 Ki 2
ZGBSEJYQXDWFRF 9.4 Ki 2
MYLRUMTYZFICQR 9.4 IC50 3
HYJRTXSYDAFGJK 9.4 IC50 5
SXLRCJRTHFTCEE 9.4 Ki 2
DDAFFKQDEBQDHP 9.3 Kd 3
XXWOCVWJOICKHA 9.3 Kd 5
PEOXDNXZHVLPEP 9.3 Ki 3
ZNXQAFLLESPBNZ 9.3 Ki 5
AIZMFPJJDXEQKC 9.3 Ki 4
OFTJLQGRWRVUFL 9.3 Ki 4
PMSLDIHTDBABLG 9.3 IC50 3
ZYYNDNILFMUVTL 9.3 IC50 2
GGUFXFJFGJKSMI 9.3 Ki 2
SPCFAZXKBQPYBW 9.3 Kd 3
VUXFZBTYCXVWMW 9.3 Ki 2
WRQYCBDVBKXRPN 9.3 Ki 2
WWLARDYNKWZLHG 9.3 Ki 2
XJHGFZGUOALOCT 9.3 IC50 2
ZGAIDOGAKIQCJU 9.3 IC50 3
ZPWHCUCZMYCWNB 9.3 Ki 2
NEAHJXCOGMHPKA 9.3 Ki 2
NPDFULBIQZLKSB 9.3 Ki 4
SSQJHXZOEJZLAK 9.3 Ki 4
LVPIEYVPDBYBIT 9.3 Ki 3
RKUNBYITZUJHSG 9.3 Ki 5
XWZQPFIZAGITHQ 9.3 Ki 4
UBDKDGUJMUUUTQ 9.3 IC50 2
ZMCUJOGARKOVLZ 9.3 Ki 3
UBDKDGUJMUUUTQ 9.3 IC50 2
WCMVSMOIDILBOJ 9.2 Ki 5
ZPUIFOBXUIMYGP 9.2 IC50 3
CNWBYOPCIWGBPG 9.2 IC50 3
DIQXIWJNNCBKDZ 9.2 IC50 3
DKTWKXDPNDGOBL 9.2 IC50 2
DKTWKXDPNDGOBL 9.2 IC50 2
2D structure