Target Details
UniProt ACP20309
Gene SymbolCHRM3
Protein NameMuscarinic acetylcholine receptor M3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,440
  • Clinical molecules 32
  • Avg pChEMBL 7.8
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (1,440)
InChIKey pChEMBL Type Targets Clinical
OPPIYDDWZLYOPO 9.6 Ki 2
PMSLDIHTDBABLG 9.6 IC50 3
QCYOIEZHUQHFEJ 9.6 Ki 3
SRPRVOSLJVWJOJ 9.6 Ki 2
UCBXWLPRAVDTBU 9.6 Ki 5
UXEIWFVTAFVRHB 9.6 Ki 2
VDLFTAVQHMFQHW 9.6 Ki 2
WDKPUEPPLMNTGG 9.6 Ki 2
ZBEWUYNNNHETOS 9.6 Kd 3
ZGBSEJYQXDWFRF 9.6 Ki 2
RKUNBYITZUJHSG 9.6 Ki 5
WOMCGBFNBSIIEA 9.6 Ki 5
AFCWMWBOATWMJV 9.6 Ki 24
FPCBWBHSQIVWBN 9.6 Ki 3
OLYUOAVKDLVFLJ 9.5 Ki 5
CNPFYHSXAKKLOF 9.5 Ki 4
IMXGJEUXZLJUBM 9.5 IC50 2
JEEPGBSHIOBHQN 9.5 IC50 3
OPRQRGHVAAWHMO 9.5 IC50 2
ZUICJRIEMALFLN 9.5 IC50 3
ASMXXROZKSBQIH 9.5 IC50 5
MYLRUMTYZFICQR 9.5 IC50 3
VWBQUAMKHIBZSG 9.5 Ki 5
BPBDCOLBZYWXHD 9.5 Ki 24
CORHJTPMSJPFRV 9.5 Ki 2
DENKZAPZMPGKBS 9.5 Ki 2
GTJTVOBMGAUNFW 9.5 Ki 2
HPUTUJYQVKLZFM 9.5 Ki 2
KSEMPLIGOKISPC 9.5 Ki 2
OEXHQOGQTVQTAT 9.5 Ki 5
OIVUQKJVYIDTLN 9.5 Ki 2
PUJDPHOMQUAXSL 9.5 Ki 2
QFRVKHZZZPVSQW 9.5 Ki 2
XELSLLUJXUXNOB 9.5 Ki 2
CZFARYRCUMIUSD 9.5 IC50 2
KQCRPVVAJACIHG 9.5 Ki 3
NHSNVFUDXZEPFP 9.5 Ki 2
YCNOXWXLGBFFOF 9.5 Ki 2
LATYFBCANWEEBS 9.5 Ki 3
WCMVSMOIDILBOJ 9.5 Ki 5
STCLPZTXPMXQOZ 9.5 Ki 3
YPVDFQGJKYMNFO 9.4 Ki 2
NTARVXTWEZJQNE 9.4 IC50 2
UVVAXSWZJPKXLR 9.4 Ki 3
IBNSRKXSITXGAZ 9.4 IC50 2
OLZRBZLJTKELRL 9.4 Ki 4
BHAUVKSALKMKRU 9.4 Ki 4
DKABYCZEFMBXSO 9.4 Ki 4
OEXHQOGQTVQTAT 9.4 Ki 5
OUUOAZNFNHOROT 9.4 Ki 3
2D structure