Target Details
UniProt ACP20309
Gene SymbolCHRM3
Protein NameMuscarinic acetylcholine receptor M3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,440
  • Clinical molecules 32
  • Avg pChEMBL 7.8
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (1,440)
InChIKey pChEMBL Type Targets Clinical
MYPZCEVGYLOQEB 11.0 Ki 2
UCQJOURWRWSNPF 11.0 Ki 2
ZOZCBLGQKDOWFZ 11.0 Kd 3
SFYPHKLFRMGESL 10.9 Ki 2
VIOKBNDQBQFHDH 10.9 Kd 3
LERNTVKEWCAPOY 10.8 Ki 6
KWNNFRFNOLSRJT 10.8 Kd 3
BEAHWTUOXGWPGA 10.7 Ki 2
MWLALRQZBOOMRW 10.7 Kd 3
CHFVEWGLPHGQML 10.3 Ki 2
LERNTVKEWCAPOY 10.3 Ki 5
NAOXUXMOYDUMFJ 10.3 Kd 3
WEFKYTFPJRTGKU 10.3 Kd 3
BKLAJZNVMHLXAP 10.2 Kd 3
FVTWTVQXNAJTQP 10.2 Kd 3
AOWQUSXFAHEKKS 10.2 Ki 2
OAWZSUHVKPQVIU 10.2 Ki 2
UUUBKRWEOPRKFC 10.2 Ki 2
WKRZFUUGOIWNNT 10.2 Ki 2
YWSIONULMMKTSJ 10.2 Ki 2
GUWDPEQJYFKDCE 10.2 Ki 3
KBNPGVPUYYZVTB 10.2 Ki 3
PRPBOUUIRMITJF 10.1 Ki 3
XXWOCVWJOICKHA 10.1 Kd 5
ZTUYXANCGWZAKE 10.1 Ki 2
FUWNRRAIDXLPKG 10.1 Ki 2
LABGCBWSNGTBPM 10.1 Ki 2
MNHIAFLMHVAZPM 10.1 Ki 3
HLWLKLSVJQAUNS 10.1 Ki 3
UKXSKSHDVLQNKG 10.1 Ki 5
JFEFOFYHVIMFRD 10.0 Kd 3
MPKFFZIONLBHKZ 10.0 Ki 2
MXCOVFAJNYVLIQ 10.0 Kd 3
PZKXTOJPCGPELH 10.0 Ki 2
WEHMQBKOLANBES 10.0 Ki 2
YYCRMTWEYYSCRD 10.0 Ki 2
MTYMLJSBEPCLGC 9.9 IC50 3
GWAMGWDJCYIREE 9.9 Kd 20
IWBMAAUPHUCYCI 9.9 Kd 20
MODBIBJHAWXYOZ 9.9 Kd 20
ZRQMUCDHVVOENY 9.9 Kd 17
WOMCGBFNBSIIEA 9.9 Ki 5
DCDOHBQTWBNVBY 9.9 Ki 2
DENKZAPZMPGKBS 9.9 Ki 2
GTJTVOBMGAUNFW 9.9 Ki 2
LERNTVKEWCAPOY 9.9 Ki 2
NVEMUJANQDPDSC 9.9 Ki 2
OAWZSUHVKPQVIU 9.9 Ki 3
OQDFIXOAMVDMRY 9.9 Ki 2
SAQVPJZBCVDTKY 9.9 Ki 2
2D structure