Target Details
| UniProt AC | P20248 |
|---|---|
| Gene Symbol | CCNA2 |
| Protein Name | Cyclin-A2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 1,415
- Clinical molecules 133
- Avg pChEMBL 7.06
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (1,415)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NPPBDFFMJNUJRY
|
7.5 | IC50 | 2 | — | |
OYWQYSATLUKKCZ
|
7.5 | IC50 | 4 | — | |
HCAPKVUYVLOOHA
|
7.5 | IC50 | 5 | — | |
DIKZCYKVEDCJAC
|
7.4 | IC50 | 3 | — | |
GZKUIKKDBXPCIY
|
7.4 | IC50 | 13 | Yes | |
HQTXGTXCDFXDLO
|
7.4 | IC50 | 3 | — | |
JSEIFJGDPNHSLS
|
7.4 | Kd | 4 | — | |
TXYKUCFACDXMFT
|
7.4 | IC50 | 7 | Yes | |
XSAQISWEGTUJBT
|
7.4 | IC50 | 7 | — | |
BLDHGAPCVONUSK
|
7.4 | IC50 | 2 | — | |
DZKFJBACCWTQSQ
|
7.4 | Kd | 4 | — | |
GSBMBRRRCWHIEM
|
7.4 | IC50 | 2 | — | |
PUNSFHAWASZDFO
|
7.4 | IC50 | 3 | — | |
RIGZCVNCFXYBEG
|
7.4 | IC50 | 11 | Yes | |
UAOIPNOTWOYAMU
|
7.4 | IC50 | 11 | Yes | |
ZEHXSPZMRLUPSR
|
7.4 | IC50 | 7 | Yes | |
ZFIVXDMTQOXNGE
|
7.4 | Kd | 4 | — | |
ATTMEZRDDPAMBY
|
7.4 | IC50 | 3 | — | |
HTRPJPBYPJZVLQ
|
7.4 | IC50 | 3 | — | |
JDLWXFAHNYGPKR
|
7.4 | IC50 | 2 | — | |
OUSFTKFNBAZUKL
|
7.4 | IC50 | 58 | Yes | |
RBAODIAUJYQMMC
|
7.4 | IC50 | 4 | — | |
SVBJNUDKKXGVHI
|
7.4 | IC50 | 5 | — | |
TVQIAQPBIDLYOL
|
7.4 | IC50 | 4 | — | |
UTSGUQQUFYMTLL
|
7.4 | IC50 | 4 | Yes | |
VPYBJHYVRIXQPO
|
7.4 | IC50 | 2 | — | |
OGSRQFDFVWCHCS
|
7.4 | Kd | 4 | — | |
QAWBPBLABQUSRL
|
7.4 | IC50 | 9 | — | |
QZEZKSMIUTYGRU
|
7.4 | IC50 | 9 | — | |
SXJKXTZFHYHUNX
|
7.4 | IC50 | 3 | — | |
SZVPDWROAQYJHW
|
7.4 | IC50 | 3 | — | |
AGPQNNSQYCHUHR
|
7.4 | IC50 | 5 | — | |
BIKJIRVRDFVXQG
|
7.4 | IC50 | 6 | — | |
GHBWBLLGGANTFE
|
7.4 | IC50 | 3 | — | |
MTIKFQKFTRIHCE
|
7.4 | IC50 | 3 | — | |
OMQDZRXQVJBWCY
|
7.4 | IC50 | 4 | — | |
OXYPRCRPNQCMEQ
|
7.4 | IC50 | 5 | — | |
VNXRLRWKODRZOV
|
7.4 | Kd | 4 | — | |
XDEIHTNJRRVHEQ
|
7.4 | IC50 | 5 | — | |
PJIPYWGIYRUKIG
|
7.4 | Ki | 8 | — | |
BCKLVLDQAAHMQR
|
7.4 | Ki | 9 | — | |
HQLLBNGXUFAPMX
|
7.4 | IC50 | 2 | — | |
MCFCYLCLAYXQIZ
|
7.4 | Ki | 9 | — | |
SQUNOCMDMIQIQK
|
7.4 | IC50 | 10 | — | |
BGPUFSMDGGQOIE
|
7.4 | Ki | 9 | — | |
GBUFGAHGZPUUTQ
|
7.4 | Kd | 4 | — | |
HUNWQLBOLVYRMW
|
7.4 | IC50 | 11 | — | |
UIEXDKQSWATHMD
|
7.4 | IC50 | 3 | — | |
WVRPZYQKQWOMIH
|
7.4 | Ki | 8 | — | |
YRFOQHHFWYWAST
|
7.4 | IC50 | 22 | — |