Target Details
| UniProt AC | P20248 |
|---|---|
| Gene Symbol | CCNA2 |
| Protein Name | Cyclin-A2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 1,415
- Clinical molecules 133
- Avg pChEMBL 7.06
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (1,415)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ITRNHZPVFGOWGQ
|
7.6 | IC50 | 3 | — | |
KMHNZVWSMBCPMT
|
7.6 | IC50 | 8 | — | |
QNUKRWAIZMBVCU
|
7.6 | IC50 | 17 | Yes | |
CDNCNMWWSCRJGY
|
7.5 | IC50 | 3 | — | |
HFEVNTGRPXCJIM
|
7.5 | IC50 | 6 | — | |
LEDNSKJDSVXHBN
|
7.5 | IC50 | 3 | — | |
OYBUHXCVUFCTQD
|
7.5 | IC50 | 3 | — | |
CEIJSVLEARLWRF
|
7.5 | IC50 | 13 | — | |
CFVWLSFPWIECRQ
|
7.5 | Ki | 9 | — | |
DSYAGVYPTCYGKP
|
7.5 | IC50 | 5 | — | |
NTUSSPZSLWLBQF
|
7.5 | IC50 | 3 | — | |
ORKSQVXJLGIROJ
|
7.5 | IC50 | 4 | — | |
PUXCYCHNNDMPTI
|
7.5 | IC50 | 3 | — | |
SBNNOXYSSSCMJX
|
7.5 | IC50 | 6 | — | |
XRHXLPUHGOTIJG
|
7.5 | IC50 | 3 | — | |
YPRFZGADERCJFT
|
7.5 | IC50 | 3 | — | |
ZRKZVQWEOWMPPZ
|
7.5 | IC50 | 3 | — | |
SPKWRLBKVPRPMT
|
7.5 | IC50 | 9 | — | |
ABDGGOBNHQMXIJ
|
7.5 | IC50 | 3 | Yes | |
AMPGTDPLFIQJLI
|
7.5 | IC50 | 3 | — | |
BOLOCLITWRGHFA
|
7.5 | IC50 | 6 | — | |
CDEIEGNYDSWLCD
|
7.5 | IC50 | 3 | — | |
CHSPOGGCOKIJJT
|
7.5 | IC50 | 3 | — | |
CSLGOZXFBHTYAA
|
7.5 | Ki | 9 | — | |
LOYSCNBYDPTSAA
|
7.5 | IC50 | 10 | — | |
LRKDOQPVSVUIPK
|
7.5 | IC50 | 3 | — | |
NSLNFDFRWNVNFZ
|
7.5 | IC50 | 3 | — | |
ZXKIYROXQGLAMR
|
7.5 | IC50 | 2 | — | |
BGFIVDZJUZNYNB
|
7.5 | IC50 | 3 | — | |
MRLPFDAKEJSGRI
|
7.5 | IC50 | 3 | — | |
PFBMBYULIZGMBA
|
7.5 | IC50 | 4 | — | |
QUUWFJNPVOBROF
|
7.5 | Kd | 4 | — | |
VJFZHLXFXHOTLG
|
7.5 | IC50 | 4 | — | |
ANZDEYYSOIFTCU
|
7.5 | Ki | 8 | — | |
AOJLBKYLAVRMQT
|
7.5 | IC50 | 3 | — | |
BFKUCEFNAQZJSZ
|
7.5 | IC50 | 2 | — | |
NQQUFCAHMNCUIZ
|
7.5 | IC50 | 3 | — | |
CUVLPOCXZYLQBD
|
7.5 | IC50 | 6 | — | |
YUJQCKBKJPDNIA
|
7.5 | IC50 | 4 | — | |
HPIIKSFGPMWKJM
|
7.5 | IC50 | 5 | — | |
HSOAJSRVFMRIRY
|
7.5 | IC50 | 3 | — | |
JKLNMYJBWWAZSO
|
7.5 | IC50 | 3 | — | |
XMDLNBHGNQECLZ
|
7.5 | IC50 | 4 | — | |
FLXKJXLZBWOYGN
|
7.5 | IC50 | 3 | — | |
LVJZZDNNQXAXPX
|
7.5 | Ki | 7 | — | |
MREGZYIBCQDRSY
|
7.5 | IC50 | 4 | — | |
NUDSGDYZHKNNPW
|
7.5 | IC50 | 3 | — | |
IHBOEHLUIBMBMY
|
7.5 | IC50 | 7 | Yes | |
INHALJGLLQNZLN
|
7.5 | Ki | 5 | — | |
MXLJQTVDWFSRDC
|
7.5 | IC50 | 3 | — |