Target Details
| UniProt AC | P20248 |
|---|---|
| Gene Symbol | CCNA2 |
| Protein Name | Cyclin-A2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 1,415
- Clinical molecules 133
- Avg pChEMBL 7.06
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (1,415)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OZMNMGRHACMSBT
|
7.7 | IC50 | 6 | Yes | |
PGGLRAWFUJMQBN
|
7.7 | Kd | 4 | — | |
SYBNWJLVMPEJGJ
|
7.7 | IC50 | 3 | — | |
UICKKEXHGQXSQJ
|
7.7 | Kd | 4 | — | |
UOLGGWWZSJIIHY
|
7.7 | IC50 | 3 | — | |
VFTAGJFGUKLKPJ
|
7.7 | Ki | 7 | — | |
ZCUPTZASSFWMPJ
|
7.7 | IC50 | 3 | — | |
AKGTYSYXMRZPBV
|
7.7 | IC50 | 9 | — | |
KGKZQGKYJDNBDP
|
7.7 | IC50 | 2 | — | |
AZPRRIBSKMOFDL
|
7.7 | Ki | 8 | — | |
BUVPYHQHZUQYBS
|
7.7 | IC50 | 7 | Yes | |
LUHGNQLUGTWNCL
|
7.7 | Ki | 12 | — | |
PUBSTGHGWFWUTL
|
7.7 | Ki | 4 | — | |
QBZJXRZGTAPTRK
|
7.7 | IC50 | 4 | — | |
XCIGDMLFQKYLKU
|
7.7 | Ki | 4 | — | |
XZQBJKPCLITHDB
|
7.7 | Ki | 12 | — | |
YEGUKZXZMMRPDN
|
7.7 | Kd | 4 | — | |
ZMMQBFMCEGTJCX
|
7.7 | IC50 | 2 | — | |
AUTIVJGNZXILJJ
|
7.6 | IC50 | 3 | — | |
DUZMNSPOOJGCPL
|
7.6 | IC50 | 3 | — | |
FAMCONSWGPBLET
|
7.6 | IC50 | 4 | — | |
HCLVUOIGTCCQQB
|
7.6 | IC50 | 3 | — | |
IRQVBNQXTXFQTM
|
7.6 | IC50 | 3 | — | |
KKNXJZMTIWJEEF
|
7.6 | IC50 | 4 | — | |
PZERAHOWFARGGG
|
7.6 | Kd | 4 | — | |
ZPKXDHHDZZKMKI
|
7.6 | IC50 | 6 | — | |
CRZXYCJOVDIWGP
|
7.6 | IC50 | 4 | — | |
FNRJTMUROZAOIB
|
7.6 | IC50 | 4 | — | |
GNJFUEMVZYQNNS
|
7.6 | IC50 | 4 | — | |
IUVOVXQLMSRQDH
|
7.6 | IC50 | 3 | — | |
LBVIZFWUIQSZHP
|
7.6 | IC50 | 10 | — | |
PSWOMNFIVDHMDM
|
7.6 | IC50 | 6 | — | |
PWMQUOFEZWCTAE
|
7.6 | IC50 | 3 | — | |
VQNXOAVFMIVTAT
|
7.6 | IC50 | 7 | Yes | |
YOPGDOJJGFKDRC
|
7.6 | IC50 | 3 | — | |
GQDHKYZSKSDSNQ
|
7.6 | IC50 | 3 | — | |
NJXVAAHYUFZELV
|
7.6 | IC50 | 6 | — | |
SXVVQLGGDQUNKQ
|
7.6 | IC50 | 5 | — | |
TZBRTWANJDQXNF
|
7.6 | IC50 | 3 | — | |
VLBVJPDXCSRGGN
|
7.6 | IC50 | 3 | — | |
VZNOTQXWDLWJSQ
|
7.6 | IC50 | 2 | — | |
XNKBKFNLOYVTSF
|
7.6 | IC50 | 3 | — | |
HXOTVSDBXJSUKD
|
7.6 | IC50 | 4 | — | |
HFTMAKGAOQSXPI
|
7.6 | IC50 | 3 | — | |
NUXMDKWZVUQHTP
|
7.6 | IC50 | 3 | — | |
OHPGMZBNBHNXPV
|
7.6 | IC50 | 4 | — | |
XSJWROYTYXTZKU
|
7.6 | IC50 | 3 | — | |
AGRGOPGRMMWYAC
|
7.6 | IC50 | 3 | — | |
AGRGOPGRMMWYAC
|
7.6 | IC50 | 3 | — | |
HMUYSTSHIXJVRO
|
7.6 | IC50 | 5 | — |