Target Details
| UniProt AC | P20248 |
|---|---|
| Gene Symbol | CCNA2 |
| Protein Name | Cyclin-A2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 1,415
- Clinical molecules 133
- Avg pChEMBL 7.06
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (1,415)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GJHVXBPCYTULDM
|
7.9 | IC50 | 4 | Yes | |
NYRVLHGVDPPWJS
|
7.9 | Ki | 5 | — | |
VIHUAIODGTUZLN
|
7.9 | IC50 | 3 | — | |
XUGUDFCFRSMZSF
|
7.9 | IC50 | 3 | — | |
VUGJTXJFAXFOGN
|
7.9 | IC50 | 2 | — | |
FOIWJMGHUDACNX
|
7.9 | IC50 | 3 | — | |
GAFYDJGFHJBXQQ
|
7.9 | Ki | 9 | — | |
KRKQVGZXTNLQSV
|
7.9 | IC50 | 9 | Yes | |
NOQYGKAHNPQBEW
|
7.9 | IC50 | 3 | — | |
OUFGAEIXDBKNPC
|
7.9 | IC50 | 3 | — | |
RLTFKHPSPUGIRA
|
7.9 | IC50 | 3 | — | |
VXBAJLGYBMTJCY
|
7.9 | IC50 | 34 | Yes | |
WAJZMHFJIYMYOJ
|
7.9 | IC50 | 3 | — | |
ZUSSYTUFZXQWGO
|
7.9 | IC50 | 4 | — | |
OEHHKRVHXQAAQT
|
7.9 | IC50 | 3 | — | |
BXSSOAIGLMVYQR
|
7.8 | Ki | 8 | — | |
JZIDYKXHTRKVEP
|
7.8 | IC50 | 5 | — | |
LVELIXLMLUGJEH
|
7.8 | IC50 | 4 | — | |
NCKHSDFHCYCSFF
|
7.8 | IC50 | 3 | — | |
NCSLRHGXEKHUGV
|
7.8 | IC50 | 3 | — | |
NVMFUMAPEQWKHK
|
7.8 | IC50 | 2 | — | |
PSNUTPHNERQRHY
|
7.8 | Ki | 4 | — | |
RNNCVRNBQXSBEN
|
7.8 | IC50 | 3 | — | |
UOSAKCKTUUCAQF
|
7.8 | IC50 | 3 | — | |
VMSMVRDDPGJMQF
|
7.8 | IC50 | 5 | — | |
YRWDEKPEPUVMIZ
|
7.8 | IC50 | 3 | — | |
DKTHMZUTCUNQAZ
|
7.8 | IC50 | 5 | — | |
OYYOJGJYZPMUHT
|
7.8 | IC50 | 4 | — | |
CSRROEXIZXVOPU
|
7.8 | IC50 | 4 | — | |
DZFYFXAPZWMNAS
|
7.8 | IC50 | 3 | — | |
FZHFVGHEAYFGKQ
|
7.8 | IC50 | 4 | — | |
KGLRLXMTNCPNET
|
7.8 | IC50 | 3 | Yes | |
OLUKILHGKRVDCT
|
7.8 | IC50 | 44 | Yes | |
RVGFQABNRSQREF
|
7.8 | IC50 | 3 | — | |
SYCCUDVKTARJAW
|
7.8 | IC50 | 3 | — | |
XLZANAXESDHDPY
|
7.8 | Ki | 8 | — | |
XQNOWBKVNDCBHZ
|
7.8 | IC50 | 4 | — | |
WOMLKCSHPRCING
|
7.8 | IC50 | 2 | — | |
FFVIVTCGXATTRT
|
7.8 | IC50 | 4 | — | |
GBUFGAHGZPUUTQ
|
7.8 | Kd | 4 | — | |
GRJMSFULANHLPW
|
7.8 | IC50 | 3 | — | |
MEPJUBFFZUKRSK
|
7.8 | Kd | 4 | — | |
MUPFEKGTMRGPLJ
|
7.8 | IC50 | 3 | — | |
NFTJDXGFOUFNKG
|
7.8 | IC50 | 4 | — | |
RSCVJZXCKTYHOT
|
7.8 | IC50 | 3 | — | |
SMWJYKRUKGMKJV
|
7.8 | IC50 | 11 | — | |
WHDHBZVTAJDTDO
|
7.8 | IC50 | 10 | — | |
XBCKUDPRGSZKAN
|
7.8 | IC50 | 4 | — | |
YANIJISPXQRULY
|
7.8 | Ki | 8 | — | |
ZIPADUJETRCYRU
|
7.8 | Ki | 4 | — |