Target Details
| UniProt AC | P20248 |
|---|---|
| Gene Symbol | CCNA2 |
| Protein Name | Cyclin-A2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 1,415
- Clinical molecules 133
- Avg pChEMBL 7.06
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (1,415)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XUCCYQOJRXEQCN
|
8.1 | Ki | 5 | — | |
BRYMZSSAIDEFEM
|
8.1 | IC50 | 4 | — | |
LXQRFMWTQCXDPP
|
8.1 | IC50 | 4 | — | |
DRYXVGHAKVVZFL
|
8.1 | IC50 | 3 | — | |
HCEVZIBGQRWFCG
|
8.1 | IC50 | 9 | — | |
HUXYBQXJVXOMKX
|
8.1 | IC50 | 28 | — | |
HZRJYORBAMJSIQ
|
8.1 | IC50 | 7 | Yes | |
ILYYGWWTDBOGTR
|
8.1 | IC50 | 3 | — | |
MYMHNTVTLZQVKZ
|
8.1 | IC50 | 7 | Yes | |
POXFFLVULXWZDC
|
8.1 | IC50 | 4 | — | |
QWTLNMRLRGDLQY
|
8.1 | IC50 | 3 | — | |
XZDHZYQSEWOJPD
|
8.1 | IC50 | 3 | — | |
XCBJCPRTHXKIAE
|
8.1 | IC50 | 3 | — | |
NFTJDXGFOUFNKG
|
8.1 | IC50 | 16 | — | |
AJXGHWYKQWIXBJ
|
8.1 | IC50 | 4 | — | |
MDPQZSCXKLJMQD
|
8.1 | IC50 | 7 | Yes | |
QKWMIPQJODDALR
|
8.1 | IC50 | 3 | — | |
WDHVWMXOJHHBQJ
|
8.1 | IC50 | 3 | — | |
WTJYXNCBJUYEKS
|
8.1 | IC50 | 3 | — | |
YUZFQJVRZIQCGL
|
8.1 | IC50 | 3 | — | |
YQOZFMRCEONJEU
|
8.0 | IC50 | 13 | — | |
BDIRGDVPAXGXBM
|
8.0 | Kd | 4 | — | |
DWHVZCLBMTZRQM
|
8.0 | IC50 | 6 | — | |
FHLJVZAGXXPSEH
|
8.0 | IC50 | 2 | — | |
HLJHKVNZSXUMIL
|
8.0 | IC50 | 4 | — | |
JJAGEMUIGMCACE
|
8.0 | IC50 | 4 | — | |
JPAVVQWCECWANY
|
8.0 | IC50 | 3 | — | |
KTERAHWGWLFDLN
|
8.0 | IC50 | 3 | — | |
MANZCDIQWXSESD
|
8.0 | IC50 | 3 | — | |
MBFRPRCYZAVISU
|
8.0 | IC50 | 4 | — | |
NCXCJSWWOBAQCH
|
8.0 | IC50 | 4 | — | |
OHZVXKQYXMVYBA
|
8.0 | IC50 | 4 | — | |
PYFVXOCGURDMHR
|
8.0 | IC50 | 3 | — | |
QFKHYTSJLGIBEQ
|
8.0 | IC50 | 4 | — | |
QVMLLKMJKQGGDX
|
8.0 | IC50 | 3 | — | |
XTBUCBOROGHGGY
|
8.0 | IC50 | 4 | — | |
ZOLPUEOXQAILTM
|
8.0 | Ki | 9 | — | |
HUKJRDDXELSRFT
|
8.0 | IC50 | 4 | — | |
BKVJIBAADPVALB
|
8.0 | Ki | 5 | — | |
GGEWEQJWGGJUHO
|
8.0 | IC50 | 8 | Yes | |
IOOBSCBCJCFBKU
|
8.0 | IC50 | 3 | — | |
JNMFNQYJOKDMNT
|
8.0 | IC50 | 3 | — | |
SMHOLGURUXBSTC
|
8.0 | IC50 | 3 | — | |
OWXORKPNCHJYOF
|
8.0 | IC50 | 17 | Yes | |
VZBGYKSZEPEEDD
|
8.0 | IC50 | 3 | — | |
OHNWBGGGJMOKIX
|
7.9 | IC50 | 4 | — | |
AJQWHEHMQASSNJ
|
7.9 | IC50 | 4 | — | |
BJDCORPGTMJYTL
|
7.9 | IC50 | 3 | — | |
CJDWWOZYUHVICE
|
7.9 | IC50 | 6 | — | |
CUZZHCAJGYQFDT
|
7.9 | IC50 | 3 | — |