Target Details
| UniProt AC | P20248 |
|---|---|
| Gene Symbol | CCNA2 |
| Protein Name | Cyclin-A2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 1,415
- Clinical molecules 133
- Avg pChEMBL 7.06
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (1,415)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YGZQAQIWZFMADC
|
8.7 | IC50 | 12 | — | |
YUJZDAUCYWRKAP
|
8.7 | IC50 | 3 | — | |
YZVFJIYEYQIHIP
|
8.7 | IC50 | 15 | — | |
ZYQXOZKYXADECC
|
8.7 | IC50 | 5 | Yes | |
QYLYUTQSYHCBOD
|
8.7 | IC50 | 13 | — | |
KGJVKYSVVOQPDL
|
8.6 | IC50 | 13 | — | |
FONDNEXKEYTNCS
|
8.6 | IC50 | 4 | — | |
NBSJZWFDNFWQDN
|
8.6 | IC50 | 29 | — | |
OXSBHNFOHBJSEQ
|
8.5 | IC50 | 4 | — | |
AFMWZFUPVUGJPF
|
8.5 | IC50 | 3 | — | |
AXAQVNRYNMCZCK
|
8.5 | Ki | 10 | Yes | |
BQLLLVDIZXOQJD
|
8.5 | Ki | 8 | — | |
DIASEXMEBNQQHZ
|
8.5 | IC50 | 13 | — | |
GAIOPWBQKZMUNO
|
8.5 | Ki | 13 | — | |
GKTNOVUFHDVNPA
|
8.5 | IC50 | 4 | — | |
HJKBVLZABNNRFO
|
8.5 | IC50 | 5 | Yes | |
KZKOIZXRAQJRPY
|
8.5 | Ki | 5 | — | |
LQBKAYJFACGUCC
|
8.5 | IC50 | 3 | — | |
MEKASOQEXYKAKM
|
8.5 | IC50 | 4 | — | |
OXPLZKSKLWBEIM
|
8.5 | IC50 | 8 | Yes | |
PIMQWRZWLQKKBJ
|
8.5 | IC50 | 36 | — | |
UPQKBKLECVIXJR
|
8.5 | IC50 | 12 | — | |
XVSQCPXHQMSQEO
|
8.5 | IC50 | 4 | — | |
YVRLFXOPNVVCQT
|
8.5 | Ki | 5 | — | |
ZHMRPXZRUZLCNL
|
8.5 | IC50 | 8 | Yes | |
ZOBRPBVIEUWYJR
|
8.5 | IC50 | 5 | Yes | |
GNKARCUXNWYAPQ
|
8.5 | IC50 | 5 | — | |
IREATOXCIIIDEG
|
8.5 | Ki | 4 | — | |
XQVDBOSCUDRTCQ
|
8.5 | IC50 | 4 | — | |
DTBQJHPUJVUHNS
|
8.5 | Ki | 7 | — | |
JXJHPQHLHQTQQI
|
8.5 | IC50 | 15 | — | |
ABEYZUJMIYFBTH
|
8.4 | IC50 | 3 | — | |
CMQDHVBSNXSEQY
|
8.4 | IC50 | 4 | — | |
FLIVKVQMXOAQAK
|
8.4 | IC50 | 15 | — | |
GJHHGLCAFGSVNF
|
8.4 | IC50 | 4 | — | |
HHYDLEDJMDNGIO
|
8.4 | IC50 | 3 | — | |
IYNDTACKOAXKBJ
|
8.4 | IC50 | 17 | — | |
KMVQBPWEFOSEIR
|
8.4 | IC50 | 3 | — | |
LDTOTGIFPXIEOT
|
8.4 | IC50 | 3 | — | |
MGCAXDANYPKQKY
|
8.4 | IC50 | 4 | — | |
OTPFZAVDWPCJLJ
|
8.4 | Ki | 9 | — | |
QWDLZMUWYCLKFF
|
8.4 | IC50 | 10 | — | |
SGOFFNQMBSXTRU
|
8.4 | Ki | 9 | — | |
TYSWNLQZLBRNSE
|
8.4 | IC50 | 15 | — | |
XCYGTFKOOGNUMR
|
8.4 | IC50 | 5 | Yes | |
ZLUXKRIOOANRPI
|
8.4 | IC50 | 4 | — | |
ZODJDUZBNLTRCH
|
8.4 | IC50 | 3 | — | |
OJRJASQFNLOAKZ
|
8.4 | Kd | 5 | — | |
RTXTXTCXICRIOE
|
8.4 | Kd | 4 | — | |
ZDFKJVWFYGHALK
|
8.4 | IC50 | 3 | — |