Target Details
| UniProt AC | P20248 |
|---|---|
| Gene Symbol | CCNA2 |
| Protein Name | Cyclin-A2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 1,415
- Clinical molecules 133
- Avg pChEMBL 7.06
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (1,415)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HRKCERYJQXATNH
|
7.2 | IC50 | 11 | — | |
OSWILUKXEWYOHP
|
7.2 | IC50 | 3 | — | |
HGEJNHUGVPFHIF
|
7.2 | IC50 | 3 | — | |
LRJIEZPKWFBSEJ
|
7.2 | IC50 | 6 | — | |
LRPFDZCHJQTXPT
|
7.2 | Ki | 8 | — | |
MDSUHMLXNPZZHO
|
7.2 | IC50 | 7 | — | |
MJSXSLBYCSPRHR
|
7.2 | IC50 | 10 | Yes | |
OSFZNJFOHBZGNK
|
7.2 | IC50 | 4 | — | |
PRJNNPMIUGYOST
|
7.2 | IC50 | 14 | — | |
VBWXQPUACHCVRW
|
7.2 | IC50 | 3 | — | |
YFXWYMXXKFMSOB
|
7.2 | IC50 | 3 | — | |
AIINAKYQKGXDFN
|
7.2 | IC50 | 2 | — | |
ATBAETXFFCOZOY
|
7.2 | IC50 | 39 | — | |
DDLZLOKCJHBUHD
|
7.2 | IC50 | 23 | — | |
GHLNHRXCRGGCPK
|
7.2 | IC50 | 3 | — | |
MRFIWOQUOAXZDO
|
7.2 | Ki | 5 | — | |
OTMLAWRVLMYMDF
|
7.2 | Ki | 3 | Yes | |
PMXCMJLOPOFPBT
|
7.2 | IC50 | 17 | Yes | |
PNKAKGKYAQLZIY
|
7.2 | IC50 | 4 | — | |
QUUWFJNPVOBROF
|
7.2 | Kd | 4 | — | |
UMCRTOONIKKCKZ
|
7.2 | Kd | 4 | — | |
UNSUKTMPEHFJHC
|
7.2 | IC50 | 2 | — | |
VVXLHYKOWIXRSV
|
7.2 | IC50 | 5 | — | |
WYJJUIPBAVISMJ
|
7.2 | IC50 | 7 | Yes | |
XNRIWHPUEZHUFJ
|
7.2 | IC50 | 2 | — | |
ZDSMJEWNLYMIFP
|
7.2 | IC50 | 4 | — | |
DXMZEMWEDCPBNA
|
7.2 | IC50 | 9 | Yes | |
SCFMWQIQBVZOQR
|
7.2 | IC50 | 14 | Yes | |
DUXWDMGSXRPDFV
|
7.1 | IC50 | 3 | — | |
MCJBRLXQSAUMIC
|
7.1 | Kd | 4 | — | |
SBNNOXYSSSCMJX
|
7.1 | IC50 | 6 | — | |
YIEUCLWKZPZZLL
|
7.1 | IC50 | 4 | — | |
HCWVCCMKEVZHLU
|
7.1 | IC50 | 6 | — | |
IEMIQIMEMFFPEZ
|
7.1 | IC50 | 3 | — | |
LGTNVNQWJQDILD
|
7.1 | IC50 | 5 | — | |
NTHMDBBWWNTVAZ
|
7.1 | IC50 | 5 | — | |
RJESYXNLLLQOLH
|
7.1 | IC50 | 3 | — | |
SNYJZDUOFHESPH
|
7.1 | IC50 | 4 | — | |
UVNWLDYNLOHPKC
|
7.1 | IC50 | 5 | — | |
BHBIHSQEXUFLCT
|
7.1 | IC50 | 3 | — | |
MKQHKMLZVXCNPR
|
7.1 | IC50 | 4 | — | |
XQGRRZAMCBAEKL
|
7.1 | IC50 | 4 | — | |
BTJHWCJCRJUEGO
|
7.1 | IC50 | 7 | Yes | |
DDDXJQXLEOFIHJ
|
7.1 | IC50 | 6 | — | |
DLENXRXJIRCJJB
|
7.1 | Ki | 6 | — | |
FULPDCCIDPUWGS
|
7.1 | IC50 | 4 | — | |
KLVYMYQTRZCMLE
|
7.1 | IC50 | 11 | Yes | |
KWKWTBFZIUSWFJ
|
7.1 | IC50 | 3 | — | |
MOSIOPGNCROISC
|
7.1 | IC50 | 3 | — | |
PQWACVUXFPZERA
|
7.1 | IC50 | 5 | — |