Target Details
| UniProt AC | P20248 |
|---|---|
| Gene Symbol | CCNA2 |
| Protein Name | Cyclin-A2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 1,415
- Clinical molecules 133
- Avg pChEMBL 7.06
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (1,415)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MTJJCZRPNOKRPO
|
7.3 | Ki | 4 | — | |
GJTRIRZIYRVGHG
|
7.3 | IC50 | 4 | — | |
KGMVZSJAPXYTKH
|
7.3 | IC50 | 23 | — | |
KJJMNVMUDVNVSU
|
7.3 | Ki | 5 | — | |
SVGQRDCSVDIDOX
|
7.3 | IC50 | 6 | — | |
VQWRERKTQFNERF
|
7.3 | IC50 | 8 | — | |
AFYLTDZJAWPVBM
|
7.3 | Ki | 8 | — | |
CXDAHVCYAZVNRY
|
7.3 | Ki | 5 | — | |
FPZYYCPZIIPVNT
|
7.3 | IC50 | 4 | — | |
KVXSQZZAGHGMFE
|
7.3 | IC50 | 4 | — | |
RGRWBAXPKCSYSG
|
7.3 | IC50 | 3 | — | |
SMUQLRPBIZRLKK
|
7.3 | IC50 | 4 | — | |
XHAWHVHQZTVHLI
|
7.3 | Ki | 4 | — | |
FQJFTSMSJXOYME
|
7.2 | IC50 | 3 | — | |
HAVTUEFHYMRXDG
|
7.2 | IC50 | 7 | Yes | |
HMCJMBDXHYZRRL
|
7.2 | Ki | 9 | — | |
JAOHKYAQQCWHRG
|
7.2 | Ki | 6 | — | |
KHEWMKNNKQJGHS
|
7.2 | IC50 | 2 | — | |
RSHKUDAKRMLDCT
|
7.2 | IC50 | 3 | — | |
BTKRPPLRYLYGOR
|
7.2 | IC50 | 3 | — | |
DZQHZAAIBBSMPD
|
7.2 | IC50 | 3 | — | |
HWFOUEQKCWVCBH
|
7.2 | IC50 | 3 | — | |
JNYWLVWHCGXRPJ
|
7.2 | IC50 | 4 | — | |
KPEWGEQNXTXESG
|
7.2 | IC50 | 7 | Yes | |
PGGLRAWFUJMQBN
|
7.2 | Kd | 4 | — | |
SCWFKTCRDHIMRO
|
7.2 | IC50 | 3 | — | |
YUBJEBHGGUAVPW
|
7.2 | IC50 | 3 | — | |
ISCPEDZQFVQCAM
|
7.2 | IC50 | 3 | — | |
OUCDNSRNVVOKPA
|
7.2 | IC50 | 4 | — | |
RANSINIOMGOPCF
|
7.2 | IC50 | 3 | — | |
XOLAFGHOWMROGX
|
7.2 | IC50 | 3 | — | |
BOYUIYWAXWEOCT
|
7.2 | IC50 | 3 | — | |
DTBMYSHZPNXMDE
|
7.2 | IC50 | 8 | Yes | |
PCVRDGSBSHXSIV
|
7.2 | IC50 | 4 | — | |
QXBKFUBBGBWPCJ
|
7.2 | IC50 | 8 | — | |
URWRFSMVDXZMJH
|
7.2 | IC50 | 3 | — | |
XEMJTISGDXHELX
|
7.2 | IC50 | 8 | Yes | |
DHZFLITTYGDMNK
|
7.2 | IC50 | 3 | — | |
DMXIHKQKBYZIHM
|
7.2 | IC50 | 5 | Yes | |
FCLBVILBAPMKST
|
7.2 | IC50 | 13 | — | |
PFMKIDRZHBZULH
|
7.2 | IC50 | 6 | — | |
ZZRNITRBTLLTQE
|
7.2 | IC50 | 3 | — | |
NUQPUUVUEUDBEL
|
7.2 | Ki | 4 | — | |
OKLIXNGBJODOLI
|
7.2 | IC50 | 6 | — | |
OXPCJRJHJOIZQD
|
7.2 | IC50 | 2 | — | |
BUYWCTZLOSQWIK
|
7.2 | IC50 | 2 | — | |
IQFRBBNJBIHVDS
|
7.2 | IC50 | 4 | — | |
UIAYOLLUEZBQEH
|
7.2 | IC50 | 6 | — | |
CBMDGSCTUBJWIN
|
7.2 | IC50 | 4 | — | |
GCEJQMWZAFXILZ
|
7.2 | IC50 | 3 | — |