Target Details
| UniProt AC | P20248 |
|---|---|
| Gene Symbol | CCNA2 |
| Protein Name | Cyclin-A2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 1,415
- Clinical molecules 133
- Avg pChEMBL 7.06
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (1,415)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HQELVOAHMYHJLJ
|
7.4 | Ki | 4 | — | |
KOMNQBZWMCFDTQ
|
7.4 | IC50 | 4 | Yes | |
LEKYSYXNVDOBCA
|
7.4 | IC50 | 5 | — | |
YPBVPXIBHMXSAS
|
7.4 | IC50 | 5 | — | |
DQKJGZAOXUAOIO
|
7.3 | IC50 | 3 | — | |
GRIBJJIZUIEJFG
|
7.3 | IC50 | 3 | — | |
IRXXTCIJUUOCGV
|
7.3 | IC50 | 3 | — | |
RHBXOKIMSCJPEB
|
7.3 | Ki | 4 | — | |
WJRRGYBTGDJBFX
|
7.3 | IC50 | 16 | Yes | |
YZRRSIPTHDIILM
|
7.3 | Ki | 9 | — | |
ZLNVBIGZYRPQKY
|
7.3 | IC50 | 15 | — | |
JSJVSQMHVJPNON
|
7.3 | IC50 | 5 | — | |
OQCYIOKKFGCDSR
|
7.3 | IC50 | 4 | Yes | |
ORRMXVSTILKSNY
|
7.3 | IC50 | 3 | — | |
UTBSBSOBZHXMHI
|
7.3 | IC50 | 15 | Yes | |
MTCJIHKSTBDECF
|
7.3 | IC50 | 3 | — | |
OVPNQJVDAFNBDN
|
7.3 | IC50 | 44 | Yes | |
QXVWBJROURLRIW
|
7.3 | IC50 | 11 | — | |
WPBZYJGEMAIFMZ
|
7.3 | IC50 | 3 | — | |
KGLQVHSLHDKNTQ
|
7.3 | IC50 | 4 | — | |
MYIYDTISJDJCKB
|
7.3 | IC50 | 3 | — | |
STFCTZRFHURCAL
|
7.3 | IC50 | 4 | — | |
UDYXTWRJETXAKK
|
7.3 | IC50 | 4 | — | |
UZWDCWONPYILKI
|
7.3 | IC50 | 47 | — | |
AHWMQFPWQLNDNV
|
7.3 | IC50 | 3 | — | |
BGZRPCJRWKJCDU
|
7.3 | Kd | 4 | — | |
DMTKMRCNVGYHOZ
|
7.3 | IC50 | 9 | — | |
GVUHDEMSKMOPHW
|
7.3 | IC50 | 9 | — | |
IORBEYRNTKWGRM
|
7.3 | IC50 | 4 | — | |
ITHULDOZQFKWFX
|
7.3 | IC50 | 3 | — | |
WYMXGRUKKZVBIY
|
7.3 | IC50 | 3 | — | |
CJQHODVHGDYGJK
|
7.3 | IC50 | 2 | — | |
JGNMMLNIOWYNHJ
|
7.3 | IC50 | 8 | — | |
KTIAVDWJHSVFJO
|
7.3 | IC50 | 3 | — | |
MQWYGEKTAREIIH
|
7.3 | IC50 | 4 | — | |
OOYUOUNLWCMZHC
|
7.3 | IC50 | 3 | — | |
SVBJNUDKKXGVHI
|
7.3 | IC50 | 6 | — | |
VMSMVRDDPGJMQF
|
7.3 | IC50 | 6 | — | |
YHVVVHLDNQXTEZ
|
7.3 | IC50 | 3 | — | |
ZEJXJYCOUVOWGJ
|
7.3 | IC50 | 13 | Yes | |
ACXFBDRQBQFLGH
|
7.3 | IC50 | 3 | — | |
AMTPXYFBGSXPMD
|
7.3 | IC50 | 3 | — | |
GNTSKAUZBDGNGK
|
7.3 | IC50 | 6 | — | |
JRLCFYYHBUWFDK
|
7.3 | IC50 | 3 | — | |
MMYWILWEDPWJHZ
|
7.3 | IC50 | 6 | — | |
PRSGCCUIEFHFFU
|
7.3 | IC50 | 4 | — | |
XZZOVHIAPZXMHM
|
7.3 | IC50 | 4 | — | |
GYMVEDSUJRTLGP
|
7.3 | IC50 | 3 | — | |
JNCZJPCSDVTXED
|
7.3 | Ki | 4 | — | |
KKCXFNXPIIHRJW
|
7.3 | IC50 | 3 | — |