Target Details
| UniProt AC | P20142 |
|---|---|
| Gene Symbol | PGC |
| Protein Name | Gastricsin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07966 (A1_Propeptide) PF00026 (Asp) |
Summary
- Multi-target molecules 18
- Clinical molecules 0
- Avg pChEMBL 6.65
Active Molecules (18)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MQDDTALXSBQTQP
|
9.1 | Ki | 5 | — | |
YTIOGZLHYJDYTK
|
8.1 | Ki | 5 | — | |
BDYFZQDNIIZQQW
|
8.1 | Ki | 5 | — | |
SXQPECMJHHMDFO
|
7.9 | Ki | 5 | — | |
DVRJOUXWYVOMLR
|
7.7 | Ki | 5 | — | |
UFJYUSGISGEOOF
|
7.0 | Ki | 3 | — | |
GMHADIRIDUBUJL
|
6.0 | IC50 | 2 | — | |
GMHADIRIDUBUJL
|
6.0 | IC50 | 3 | — | |
JNBVLGDICHLLTN
|
6.0 | IC50 | 3 | — | |
KJQYIOYOHBXLEG
|
6.0 | IC50 | 4 | — | |
LUFWCAAWWRWIEJ
|
6.0 | IC50 | 2 | — | |
NFXWMRPSLAAALF
|
6.0 | IC50 | 4 | — | |
ODEIJAFXYALBOH
|
6.0 | IC50 | 3 | — | |
PRTZELVVYWACOX
|
6.0 | IC50 | 4 | — | |
RPMSJAUJPZIRMH
|
6.0 | IC50 | 3 | — | |
UVZNGTDEZCYVKR
|
6.0 | IC50 | 2 | — | |
ZFZUCSZEDBBENP
|
6.0 | IC50 | 4 | — | |
ZFZUCSZEDBBENP
|
6.0 | IC50 | 4 | — |