Target Details
| UniProt AC | P20083 |
|---|---|
| Gene Symbol | parE |
| Protein Name | DNA topoisomerase 4 subunit B |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 17
- Clinical molecules 0
- Avg pChEMBL 7.56
Active Molecules (17)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YTFKJABGFFQSEZ
|
8.5 | IC50 | 2 | — | |
IDALGTCHRLCQSK
|
8.4 | IC50 | 2 | — | |
MBCOBCDFYMQNQZ
|
8.4 | IC50 | 2 | — | |
MFKOUFLQPFIPBG
|
8.1 | IC50 | 2 | — | |
RSCJTJIKINXWDW
|
8.1 | IC50 | 2 | — | |
SZIOCYHUCPYPPG
|
8.0 | IC50 | 2 | — | |
JIYXQJVMEKXTDD
|
7.9 | IC50 | 2 | — | |
XRACSVMFYBESAS
|
7.8 | IC50 | 2 | — | |
KOVLKWGJIYFSRO
|
7.7 | IC50 | 2 | — | |
UCFIUPFZVAQTSV
|
7.6 | IC50 | 2 | — | |
WGQVVXSEZNKYIF
|
7.6 | IC50 | 2 | — | |
JETKTBLDFMGAOL
|
7.6 | IC50 | 2 | — | |
GFCYSWOAOCSVFR
|
7.3 | IC50 | 2 | — | |
TVZISUHTUGEDEK
|
6.7 | IC50 | 2 | — | |
OHKRUIKTNKYKGG
|
6.4 | IC50 | 2 | — | |
GLNFAHNABSNEAM
|
6.2 | IC50 | 2 | — | |
UNPWBBYTMMYTPY
|
6.1 | IC50 | 3 | — |