Target Details
| UniProt AC | P20035 |
|---|---|
| Gene Symbol | LACZ |
| Protein Name | Hypoxanthine-guanine-xanthine phosphoribosyltransferase |
| Organism | Plasmodium falciparum (isolate FCR-3 / Gambia) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00156 (Pribosyltran) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 7.09
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QYVPBNMGNCACHL
|
9.2 | Ki | 2 | — | |
APDUDHYPFAMPGN
|
8.0 | Ki | 3 | — | |
APDUDHYPFAMPGN
|
7.2 | Ki | 2 | — | |
KDWYBFCNTYIRFX
|
7.0 | Ki | 2 | — | |
OSIWAKYTBPSMMK
|
7.0 | Ki | 2 | — | |
ZBCWHJNHJJUGMA
|
7.0 | Ki | 2 | — | |
IVBKXHITGSVPFM
|
6.7 | Ki | 2 | — | |
JPFXXOOGZIRDPS
|
6.7 | Ki | 3 | — | |
MXUMOEQVYHYPGP
|
6.7 | Ki | 2 | — | |
TWGQTNPDFLDXBY
|
6.7 | Ki | 3 | — | |
JGCOPSLIOMTBDT
|
6.5 | Ki | 3 | — | |
BDQWSUFOTXTHGI
|
6.3 | Ki | 2 | — |