Target Details
| UniProt AC | P19525 |
|---|---|
| Gene Symbol | EIF2AK2 |
| Protein Name | Interferon-induced, double-stranded RNA-activated protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00035 (dsrm) PF00069 (Pkinase) |
Summary
- Multi-target molecules 27
- Clinical molecules 3
- Avg pChEMBL 6.46
KEGG Pathways (11)
Associated Diseases (2)
Active Molecules (27)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KWVSNBQCQKQRHX
|
7.2 | IC50 | 3 | — | |
YLCFOHVAOBLAIK
|
7.1 | IC50 | 14 | — | |
HFOKVVVCWLIUBP
|
7.0 | IC50 | 3 | — | |
NXWXUDHOUKWAQU
|
6.9 | Kd | 16 | — | |
UIARLYUEJFELEN
|
6.9 | Kd | 289 | Yes | |
APPXQUDJLJXULP
|
6.8 | IC50 | 47 | — | |
XTCSSXNPALQZJQ
|
6.8 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
6.7 | Kd | 220 | — | |
NMEUKWOOQOHUNA
|
6.6 | IC50 | 6 | — | |
SAYGKHKXGCPTLX
|
6.6 | IC50 | 4 | Yes | |
KWZXRCBCAYLKPI
|
6.5 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
6.4 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.4 | Kd | 213 | — | |
QAEKSWBVYBVLNO
|
6.4 | IC50 | 5 | — | |
DGECBIQUJWBSOF
|
6.4 | IC50 | 3 | — | |
XQVVPGYIWAGRNI
|
6.3 | Kd | 34 | — | |
HTYLSAJYCQVPBD
|
6.3 | IC50 | 3 | — | |
DDLZLOKCJHBUHD
|
6.2 | IC50 | 23 | — | |
OLOJSTRISMGUEK
|
6.2 | IC50 | 5 | — | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
SIXVRXARNAVBTC
|
6.2 | IC50 | 12 | — | |
PRWSIEBRGXYXAJ
|
6.0 | IC50 | 4 | — | |
YABJJWZLRMPFSI
|
6.0 | Kd | 34 | — | |
LIGGMBSSOOVGAE
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |