Target Details
| UniProt AC | P18858 |
|---|---|
| Gene Symbol | LIG1 |
| Protein Name | DNA ligase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF04679 (DNA_ligase_A_C) PF01068 (DNA_ligase_A_M) PF04675 (DNA_ligase_A_N) |
Summary
- Multi-target molecules 31
- Clinical molecules 0
- Avg pChEMBL 8.14
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (31)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HEIXLGZCGUTTNY
|
9.5 | IC50 | 3 | — | |
SEFMBCXQEYFZNK
|
9.1 | IC50 | 2 | — | |
GOKPISPQPCIBMS
|
8.9 | IC50 | 2 | — | |
AJTFTOJFTFVQHK
|
8.9 | IC50 | 3 | — | |
ONDWZFFDWRKXKE
|
8.8 | IC50 | 2 | — | |
QZIJGRWYLYQBLO
|
8.7 | IC50 | 2 | — | |
OOPSZFOFVBJXMF
|
8.6 | IC50 | 3 | — | |
NPLDDPZWNXUZQF
|
8.6 | IC50 | 3 | — | |
ILOIOIGZFHGSMS
|
8.5 | IC50 | 5 | — | |
IVBGIXDVHGYNIG
|
8.5 | IC50 | 2 | — | |
VAYUMGOSGZBSMF
|
8.5 | IC50 | 2 | — | |
ZPFMBPVMRCIDBP
|
8.3 | IC50 | 2 | — | |
STSOBNCCLHCLCI
|
8.3 | IC50 | 2 | — | |
UNQRPHQCMZCRIG
|
8.3 | IC50 | 2 | — | |
FBSDLZAMUQFBSX
|
8.2 | IC50 | 2 | — | |
RGBFZMIPBWNGPE
|
8.2 | IC50 | 2 | — | |
ODQCXALXZCGYKU
|
8.2 | IC50 | 2 | — | |
JPUOUZLSBPJXEV
|
8.2 | IC50 | 2 | — | |
NWUNIVMFVYNPEW
|
8.2 | IC50 | 2 | — | |
AITFDHBROVIWGR
|
8.1 | IC50 | 2 | — | |
JFADYLNYNWJEAR
|
8.1 | IC50 | 2 | — | |
VYGSYWKKZIMLJG
|
8.0 | IC50 | 2 | — | |
BBFQYOOSPUJNBB
|
7.8 | IC50 | 2 | — | |
DOQYHNYWFHIVPS
|
7.7 | IC50 | 2 | — | |
HHCOCKSGAZJTSF
|
7.6 | IC50 | 2 | — | |
MLNUKPVTGKVHLU
|
7.6 | IC50 | 2 | — | |
NLMGKBWZZZUXAF
|
7.6 | Ki | 2 | — | |
YYMQHFDGNJKEDZ
|
7.3 | Ki | 2 | — | |
NCWGFJOHLLPNNL
|
7.2 | IC50 | 2 | — | |
KMWBCGYYQBQMCP
|
6.7 | Ki | 2 | — | |
NKOSKXJRVWVXRI
|
6.0 | IC50 | 2 | — |