Target Details
UniProt ACP18825
Gene SymbolADRA2C
Protein NameAlpha-2C adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 685
  • Clinical molecules 45
  • Avg pChEMBL 7.23
Top Co-occurrence Targets
Active Molecules (685)
InChIKey pChEMBL Type Targets Clinical
MCAGSCISRRGDGQ 7.1 Ki 3
MNMDMCKHXVHLAW 7.1 Ki 4
RCLSMBSYDRCUSB 7.1 Ki 3
RGCVKNLCSQQDEP 7.1 Ki 16
AZADEQYOIWOMER 7.1 Ki 2
MQZXNJVAUSWZRL 7.1 Ki 3
VPDYOWAJRMPOEI 7.1 Ki 3
AVVCHEPXGGYIRM 7.0 Ki 2
IHCKEJIXIYLTFT 7.0 Ki 2
JNMSRIDVZNTYJE 7.0 Ki 2
KRFMDKUGQLNZKI 7.0 Ki 3
LYKMMUBOEFYJQG 7.0 Kd 6
PNISAWOKGCKONH 7.0 Ki 4
VUTLJDGDPMZCOA 7.0 Ki 3
VDRGNAMREYBIHA 7.0 Ki 11
BETHXCLHMRGYBW 7.0 Ki 9 Yes
BSOLCASXROXPRZ 7.0 Ki 9
URKOMYMAXPYINW 7.0 Ki 27 Yes
PSVIJGBMZYPVMJ 7.0 Ki 3
UEZSUAXJWCMWEK 7.0 Kd 3
WEGLOYDTDILXDA 7.0 Ki 22
ISSSVYKMIIAPTH 7.0 Ki 3
LCPAFKZCFFLTPB 7.0 Ki 3
YMHOBZXQZVXHBM 7.0 Ki 13
MJJALKDDGIKVBE 7.0 IC50 30 Yes
ODGBUUUVMLDZBP 7.0 Ki 7
HUCJFAOMUPXHDK 7.0 Ki 8
PGGCRGAETLNAJC 7.0 Ki 11
PKXHLBVPUHXZNH 7.0 Ki 3
SYPINLPWMTYMEC 7.0 Ki 3
XGMNRALXOWECNG 7.0 Ki 3
BCCMUPQZPVRDCD 6.9 Ki 6
YEHCICAEULNIGD 6.9 Ki 20
KVWDHTXUZHCGIO 6.9 Ki 32 Yes
UFVSFWQCSISIPB 6.9 Ki 3
XDAIWLKBRMSRTM 6.9 Ki 2
IPQYPIRIGUBUAF 6.9 Ki 3
PIAONGWBRPZERV 6.9 Ki 3
IAIZHDGEGFGNMO 6.9 Ki 3
PQVQCEDGSJVHMK 6.9 Ki 9
QYCJTZDZQXSXSC 6.9 Ki 3
YAYASQTZIRSRFB 6.9 Ki 3
HIHZDNKKIUQQSC 6.9 Ki 7
IAIZHDGEGFGNMO 6.9 Ki 3
WEGLOYDTDILXDA 6.9 Ki 22
HIJHJEWMVKEUOP 6.9 Ki 3
CXQUOFVDYCOSEZ 6.8 Ki 10 Yes
MJKRYUCQHJLOIV 6.8 Ki 5
YGIWTZGEYHABOR 6.8 Ki 6
YNNUSGIPVFPVBX 6.8 Ki 24 Yes
2D structure