Target Details
UniProt ACP18825
Gene SymbolADRA2C
Protein NameAlpha-2C adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 685
  • Clinical molecules 45
  • Avg pChEMBL 7.23
Top Co-occurrence Targets
Active Molecules (685)
InChIKey pChEMBL Type Targets Clinical
ASHFKBMVCDTQQO 8.0 Ki 4
HJACXCAXDLNLEL 8.0 Ki 3
LUZRJRNZXALNLM 8.0 Ki 20
GPLGAQQQNWMVMM 8.0 Ki 3
MGQIWQQQIZXANT 8.0 Ki 3
NTHIAFXFYRUEJP 8.0 Ki 3
OSEADGVOKYGIER 8.0 Ki 3
PQXKDMSYBGKCJA 8.0 Ki 3
SNBRKKJCZXXNNL 8.0 Ki 3
RNPCOHCWKNMBRI 8.0 Ki 3
FXNNPMSELIMMHU 7.9 Ki 4
RWMIVZPIQPHMSK 7.9 Ki 3
MRBDMNSDAVCSSF 7.9 Ki 10
CQXADFVORZEARL 7.9 Ki 4
ONSCHPQYHGOIQX 7.9 Ki 6
SNKCREOVGWDJDI 7.9 Ki 3
VSWBSWWIRNCQIJ 7.9 Ki 23
ZBEZMDBAFCFGAT 7.9 Ki 6
KXSUAWAUCNFBQJ 7.9 Ki 3
VNSOQQZNVNIEMP 7.9 Kd 6
JMXRRARDLWHYJN 7.8 IC50 4
YDOTUXAWKBPQJW 7.8 IC50 13
CUHVIMMYOGQXCV 7.8 Ki 7
HCMWMLSNHRNVSJ 7.8 Ki 3
MEKSQRMXWZHFIP 7.8 Ki 13
POCXNIFHHUXWMU 7.8 Ki 3
UCAIEVHKDLMIFL 7.8 Ki 4
XMXHEBAFVSFQEX 7.8 Ki 17
OLPQNRLJYOGSGV 7.8 Ki 6
OOYTZYZXCMCMSZ 7.8 Ki 3
OSJJYEUEJRVVOD 7.8 IC50 17 Yes
DZSQSLQSMKNVBV 7.8 Ki 4
ZUXABONWMNSFBN 7.8 Ki 29
BQXXXVQLOOIBPN 7.7 Ki 3
RDAVKEYAUFGPDX 7.7 Ki 3
XGMNRALXOWECNG 7.7 Ki 3
HBMJQYDGBNSZMC 7.7 Ki 4
HIASAPHKGILEIV 7.7 Ki 2
HPMRFMKYPGXPEP 7.7 Ki 10
HXHKXXRIQOWOHI 7.7 Ki 3
NDFYRGCPDAFQDG 7.7 Ki 2
CWYDYWFZPBTTIM 7.7 Ki 3
LNYCQEZPPFYNOL 7.7 Ki 2
RSRUDTPYRBLHEO 7.7 Ki 6
AJZBPCAHQHCXMX 7.7 Ki 5
WFPUBEDBBOGGIQ 7.7 Ki 4
WKXSXFYQPCWZOS 7.7 Ki 6
IEJXVRYNEISIKR 7.7 Ki 6
KORNTPPJEAJQIU 7.7 Ki 17
CVKQUGPVDVFRAT 7.6 Ki 3
2D structure