Target Details
UniProt ACP18825
Gene SymbolADRA2C
Protein NameAlpha-2C adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 685
  • Clinical molecules 45
  • Avg pChEMBL 7.23
Top Co-occurrence Targets
Active Molecules (685)
InChIKey pChEMBL Type Targets Clinical
UCNOTTVNPRSTFW 9.2 Ki 8 Yes
WNCGPEYSCDVJNB 9.2 Ki 3
GZFYZEHGCPEJAC 9.1 IC50 4
JOAHPSVPXZTVEP 9.1 Ki 19
GYSZUJHYXCZAKI 9.1 Kd 7
KOMMMRWKUHRBSF 9.1 Ki 3
RKQFKAILJGXGRP 9.1 Ki 3
HOKCXDCTKLQEJE 9.1 Ki 3
GICQFAWDMCTLDM 9.1 IC50 4
NJTFNKZJGXSOMJ 9.1 Ki 3
HQGWKNGAKBPTBX 9.0 Ki 3
PUJAGVRPJZNJPF 9.0 IC50 4
UVEKKXRFQCNLQE 8.9 Ki 4
JWXMKFUDAOLJCY 8.9 Ki 4
FGTWZUQEDNXLLZ 8.9 IC50 4
YGAFMXXNJBOVBA 8.9 Ki 3
AKBJKOBHDJQWMB 8.9 Ki 4
FPQNWBCHCMEAKI 8.9 IC50 4
RNPCOHCWKNMBRI 8.9 Ki 3
WLWNODXEXGTHDO 8.9 IC50 4
AKZOIEBLVQLVTR 8.9 IC50 3
ZFZUYTCCHMWWTD 8.8 Ki 9
HSRPTPAPMBHRRJ 8.8 IC50 5
IXRPDYSTGHYEBR 8.8 Ki 4
LQKQCQKZRUYZOI 8.8 Ki 4
RVIXAJHMKWFIKC 8.8 Ki 3
DGXYDPJRLWCWFV 8.8 Ki 3
LWSVCEUUPRLOSZ 8.8 Ki 3
UDURNHDRCUMUOV 8.8 IC50 4
XSOUHEXVEOQRKJ 8.8 Ki 14
MUUSOYWTPTTZII 8.8 Ki 3
MUUSOYWTPTTZII 8.8 Ki 3
ZYXHQIPQIKTEDI 8.8 IC50 4
HGEYJZMMUGWEOT 8.8 Ki 17
RVRPAIWBGBVSKB 8.8 Ki 3
YWALOGYVALOLTL 8.8 Ki 3
GXZWKZAOGQRNTL 8.7 Ki 12
WDCPMDKQCCZVEW 8.7 Ki 3
WYFPZXUWZCKNMJ 8.7 Ki 3
OYOGQACTFBHTOD 8.7 Ki 3
GEBHRBBICJPJRU 8.7 Ki 3
MHPMXTGKTXJIDI 8.7 Ki 6
HNRZWHPQDGUUSO 8.7 IC50 4
CNIIGCLFLJGOGP 8.6 Ki 4
FJABWASNVHOPLU 8.6 Ki 3
ZMOPTLXEYOVARP 8.6 Ki 14 Yes
SPMYVDNOOYXROZ 8.6 Ki 3
WGLYZLZIIJTKAG 8.6 IC50 4
DLWKVBPPVYZEML 8.6 Ki 4
LEHLBTBBMZYRBK 8.6 Ki 3
2D structure