Target Details
UniProt ACP18825
Gene SymbolADRA2C
Protein NameAlpha-2C adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 685
  • Clinical molecules 45
  • Avg pChEMBL 7.23
Top Co-occurrence Targets
Active Molecules (685)
InChIKey pChEMBL Type Targets Clinical
VWIAFKHHBIYXKV 10.8 IC50 3
MWIKFEVHBBAXIQ 10.8 IC50 3
VGYOOEDZRKNLKS 10.5 Ki 3
SWDBYQPERYMOIS 10.5 IC50 3
JRDUBBHIPPPSLP 10.2 Ki 3
NCOXQFRYWWZGEM 10.0 Ki 3
UCFVOQSSWZQWNE 10.0 Ki 3
YRDASYXEOGTMQU 9.9 IC50 3
FIERHAFMRVRMDV 9.8 Ki 4
ARHWJJBPLJIHQP 9.8 Ki 4
AYMCTBRVXPCORT 9.7 Ki 3
DISVZQSFAXIOLP 9.7 Ki 3
IPLOTOHAAAUTMK 9.7 Ki 3
JBOWHEDUACRXHK 9.7 Ki 3
JCJVFLLBDXJJPW 9.7 Ki 3
JKDBLHWERQWYKF 9.7 Kd 3
JKDBLHWERQWYKF 9.7 Kd 3
JPNJJWFOEQLLSP 9.7 Ki 3
JWYUBODPEUBFLH 9.7 Ki 3
JWYUBODPEUBFLH 9.7 Ki 11
LLFVSLMMRPXQFK 9.7 Ki 3
NDIXVNRNAFQAJZ 9.7 Ki 3
UHVQVIBBKZFOBO 9.7 Ki 2
BJNQZYVNKAVYSF 9.6 Ki 6
GKDBTHSYQZTDAJ 9.6 IC50 13
WCIDBLYFACGZGW 9.6 IC50 3
WYFCRYMMLDTJAM 9.5 Ki 4
BLAVUEWHVKGIIM 9.5 Ki 3
BSOFNSGMVOMVLM 9.5 Ki 3
COPXFRMTXFPQKE 9.5 Ki 3
XGXYGEYUGTVZAR 9.5 Ki 6
YMYZKGIHGMHZDL 9.5 Ki 5
VKABNRMTNPWHBD 9.4 Ki 3
PYXVPLGVUNHGEJ 9.4 Ki 3
SYULCMQGHBLEEJ 9.4 Ki 3
PRXCUMHAHRIDJF 9.4 Ki 4
KSQAWHREGPMSBF 9.3 Ki 3
OLAGLCHGSUYVBF 9.3 Ki 3
QHCZSHHKZDDCEC 9.3 Ki 3
RJLMZCSOGDTDNJ 9.3 Ki 3
VDSXZDLUEYFJGH 9.3 Ki 4
VMLJCXYBTLCGDU 9.2 Ki 3
YMYZKGIHGMHZDL 9.2 Ki 3
RTXNZOCMRSFEID 9.2 IC50 4
WVDIRTLHBANRPM 9.2 IC50 3
BKRGVLQUQGGVSM 9.2 Ki 26 Yes
JVGBTTIJPBFLTE 9.2 Ki 16
BRKWIMBSEICBCU 9.2 IC50 4
HPNSJGWCFMHOJX 9.2 IC50 4
HQDWMIAYEGTBSF 9.2 Ki 3
2D structure