Target Details
UniProt ACP18507
Gene SymbolGABRG2
Protein NameGamma-aminobutyric acid receptor subunit gamma-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,275
  • Clinical molecules 0
  • Avg pChEMBL 7.71
Top Co-occurrence Targets
Active Molecules (1,275)
InChIKey pChEMBL Type Targets Clinical
LOZNAQDBHKVLRN 8.6 Ki 6
PPTYJKAXVCCBDU 8.6 Ki 7
XPSAGIQSESMIJK 8.6 Ki 6
GXKGSEUULCEOTM 8.6 Ki 5
IGTNDWINIZAURX 8.6 Ki 3
KDUFISFQSHXSHF 8.6 Ki 3
MFZNONRIQYSLMZ 8.6 Ki 6
SUCNRFFYZAMZJS 8.6 Ki 3
FFIJKSHMFVHCAE 8.6 Ki 3
NHAVPZBYCXDYLA 8.6 Ki 3
OKOKWNYOLUGIGN 8.6 Ki 3
OXRXBJGSNZVEPW 8.6 Ki 4
YCTZWWGYTRDQQM 8.6 Ki 3
CHIFCDOIPRCHCF 8.6 IC50 16
CHQPOBHNDRMXFK 8.6 Ki 18
QZJAEUOFNKKIJN 8.6 Ki 3
QPBUEBDNKGGQCP 8.5 Ki 3
WKYYFGMWPBWQAS 8.5 Ki 3
BKGDQBJGYREIHW 8.5 Ki 3
CVOASAXXOXOGQG 8.5 Ki 5
HSKAYWQXMCMXAQ 8.5 Ki 3
KVKYGVOAHGNAKZ 8.5 IC50 17
LENHHZQGSWCZJW 8.5 Ki 16
LPAODQAWVMEXKR 8.5 IC50 16
LZTHAJBUMOQDLU 8.5 IC50 3
NEOUOHDNZDRDNJ 8.5 IC50 16
OKGJPMZATLJSGV 8.5 Ki 6
PFJHXYJLEIZLGQ 8.5 Ki 6
QIZPCEVRKTWHIE 8.5 IC50 16
RYLDZJANGRBUGW 8.5 IC50 16
YSLDYJOGEQZLDN 8.5 Ki 3
AOZALWRGTMILIK 8.5 Ki 6
BWWQXKSOWUMHAQ 8.5 Ki 6
KSYVJHGNJMYDIQ 8.5 Ki 6
QVOYXYWXOMVGNY 8.5 Ki 4
IGANKKXNZYWZFN 8.5 Ki 3
JFONUHWYOVYDJT 8.5 Ki 3
JRCQRBJGHBZPRG 8.5 Ki 3
VMKZXEMKFBINKN 8.5 Ki 3
OJVFFZLXISLIFZ 8.5 Ki 6
VAJLZGPUVKNCRO 8.5 Ki 6
KADHNYOMTSABQA 8.4 Ki 3
WZNQGAWPCOPXOK 8.4 Ki 4
DDRXKTPRVSLWJP 8.4 Ki 3
MVBVNOZDVRVMNH 8.4 IC50 16
SJAGJFDQMIAULO 8.4 Ki 6
ZKVGHURGXXUFQB 8.4 Ki 6
IGVUOCSFSJKTDF 8.4 Ki 3
JTGPXCIJDIEQSX 8.4 Ki 4
WLHRDALLBOSVLX 8.4 Ki 6
2D structure