Target Details
UniProt ACP18507
Gene SymbolGABRG2
Protein NameGamma-aminobutyric acid receptor subunit gamma-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,275
  • Clinical molecules 0
  • Avg pChEMBL 7.71
Top Co-occurrence Targets
Active Molecules (1,275)
InChIKey pChEMBL Type Targets Clinical
KCEIOBKDDQAYCM 9.2 Ki 5
KVQKVRWATUWLAO 9.2 Ki 5
LICVBNQRZFPUHS 9.2 Ki 4
QZDWWRKBDPYMIP 9.2 Ki 6
JLCBYDSLJHLQQB 9.1 Ki 5
ISZRIZPRXUQOMU 9.1 Ki 5
BQDUNOMMYOKHEP 9.1 Ki 6
CNEHRQMKOUFFMX 9.1 Ki 3
DQKNTSFPZMVKNA 9.1 Ki 3
GXPHYMCBGKIIKN 9.1 Ki 3
ILFZZMYJRPZIPF 9.1 Ki 5
JFGUJXZLJIUVPZ 9.1 IC50 16
LYFROTHEKIFZAU 9.1 IC50 16
RYIVVNHBYBYXHF 9.1 IC50 16
SRAWBNFSMIHBEM 9.1 Ki 8
VZKRZUPJCVFVGR 9.1 IC50 16
LLHQBHOWDZNCNK 9.1 Ki 5
MTNLFTKJHWYWQV 9.1 Ki 4
JNJUWXAKLRKXII 9.1 Ki 6
DGBIGWXXNGSACT 9.1 Ki 16
LODWVHSNNGQTKI 9.1 Ki 3
XXRKXVKJMSIZSM 9.1 Ki 6
LHGSGTVATLBNGO 9.1 Ki 3
XJRDHPKTMGWJGN 9.1 Ki 6
YJZGQBGGTBIAOP 9.1 IC50 16
YLDRVNNGBACDSD 9.0 Ki 6
GPTKIASBZUGFEQ 9.0 Ki 3
JYKXGGXAKPOFML 9.0 Ki 3
PNEOQFYBCKZRBL 9.0 Ki 3
AQKFCEWRKDXGMK 9.0 Ki 16
BQWZDXNKDYRCJK 9.0 Ki 3
DVVOGWYOYHNNQP 9.0 Ki 3
FVFFDKKTXYVCCW 9.0 IC50 16
IPHSQMSRIWZULE 9.0 Ki 16
KDMMIKQMHNBKAV 9.0 Ki 17
KOVRZNUMIKACTB 9.0 IC50 17
NURMFSYNABAOFU 9.0 Ki 6
OGBTVLIUFUJHTH 9.0 Ki 5
OXDLZFDSMXMUKS 9.0 Ki 3
RKWZHLJYVXAQQP 9.0 Ki 3
VQQCPWHLJXFLOG 9.0 Ki 3
WGRVAGIQTHEEQW 9.0 IC50 16
BJYKRVMKNGJKKZ 9.0 Ki 6
JOFWLTCLBGQGBO 9.0 Ki 8
OLKUNPKISSHQBO 9.0 Ki 6
VREFGVBLTWBCJP 9.0 Ki 7
BSBLYLUAUVTSMM 9.0 IC50 16
CMRJVDJLBFKXKL 9.0 Ki 4
FYOXWZFDOADHOW 9.0 Ki 6
HZDFUJFVZWUGMH 9.0 Ki 3
2D structure