Target Details
UniProt ACP18507
Gene SymbolGABRG2
Protein NameGamma-aminobutyric acid receptor subunit gamma-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,275
  • Clinical molecules 0
  • Avg pChEMBL 7.71
Top Co-occurrence Targets
Active Molecules (1,275)
InChIKey pChEMBL Type Targets Clinical
XGJLRKVQXMSBJW 8.1 IC50 16
AYVAVBFBOCMUHW 8.0 Ki 6
CTRXOLVKJBOGRK 8.0 Ki 3
HEGJYRQUDMITRQ 8.0 Ki 6
INPSWSQUPKQGLM 8.0 Ki 3
JANXKKALWNYMDP 8.0 Ki 3
QORLMYYHZLDYOR 8.0 Ki 9
FLEQTIDRWGGTRR 8.0 Ki 7
FPJZUCHOLOKXEN 8.0 Ki 3
IXGIOXIKQZCZIK 8.0 Ki 8
PYXJKYJAFMLYMS 8.0 Ki 6
YACVJANLLKEODL 8.0 Ki 4
GPVVRPMOSQNFDF 8.0 Ki 3
KWPOKTUWXDCATM 8.0 IC50 16
YVPJMZCJVHJOFG 8.0 Ki 7
YZRXMMCBUVDBFF 8.0 Ki 6
FKXQDPHVYFMAIM 8.0 Ki 3
HQJSGBKPXYZTRN 8.0 IC50 16
JEUGTSHICBOMGA 8.0 Ki 3
MBZNSAJBODIJCK 8.0 IC50 16
RTRIMAMBTITPNP 8.0 Ki 6
UBZQMNGVBPUKCE 8.0 Ki 4
VELCIJHTXAIRCT 8.0 Ki 3
VUYWTACIDAVGNA 8.0 Ki 3
YVAHCWLEKOONFT 8.0 Ki 3
GAMSSMTVVVDEJR 8.0 Ki 4
JSDYTEOPJOVCPM 8.0 Ki 6
IBPJOIOGTFGBRO 8.0 Ki 6
YJQPSUGEFJEJIN 8.0 Ki 6
CDRADZRGYBTOKU 8.0 Ki 6
FIZTZZUELBWXAD 8.0 Ki 4
FVADWXKWYJAGND 8.0 Ki 3
HFPZDEHIDKJZSN 8.0 Ki 16
IPEQYLWHCRAOTC 8.0 Ki 6
LGGQWNKPBCAIKX 8.0 Ki 3
LMJMBPXKXWIKQK 8.0 IC50 16
NNHRCSJWUBQYQV 8.0 IC50 16
PKJGSRHYDOGGLB 8.0 Ki 17
PTJXEJYDOYCHOL 8.0 IC50 3
PZIQTZQOFYKORR 8.0 Ki 6
TWSTVDPXWQPIIM 8.0 Ki 4
UBZGCHSBAOJHLE 8.0 Ki 3
UWALHBHAIPDYBK 8.0 Ki 3
ZAKVPALBELHKFH 8.0 Ki 6
ZJQHPWUVQPJPQT 8.0 IC50 17
XDMOVRKAINVBDT 8.0 Ki 3
ZACQJMKEQBFUDN 8.0 Ki 6
CUICGHSKDSXIRX 7.9 Ki 6
FJLMOGVUSSSKEC 7.9 Ki 16
LLAKESJIQFAQJA 7.9 IC50 16
2D structure