Target Details
UniProt ACP18507
Gene SymbolGABRG2
Protein NameGamma-aminobutyric acid receptor subunit gamma-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,275
  • Clinical molecules 0
  • Avg pChEMBL 7.71
Top Co-occurrence Targets
Active Molecules (1,275)
InChIKey pChEMBL Type Targets Clinical
CGMJQQJSWIRRRL 10.1 Ki 6
JWODBROOGAIDRT 10.0 Ki 3
ORCNDQDLFHQBRB 10.0 Ki 3
KWBJTSIHFVATSO 10.0 Ki 3
LTRYPGNCHZSXSI 9.9 Ki 3
NAGYYVWENUNCDU 9.9 Ki 3
TUYGGVAJDAZCIC 9.9 Ki 3
KKXPFXBGMGQSMA 9.8 Ki 3
OWENCIOAIROJMF 9.8 Ki 3
MZFKWSFOAVBLQM 9.8 IC50 16
QUUNMICPMYIHFS 9.8 Ki 16
WDBBCFFNOHDOBT 9.7 Ki 5
GFTZCCLPKHGIAB 9.7 Ki 3
GMFQPQQGURBQLQ 9.7 Ki 3
LNPVVDKIXXYELR 9.7 Ki 3
PCLDOYFAYOCLQE 9.7 Ki 3
PPAPIXRCRCPGPU 9.7 Ki 3
RCZMTZGAJGJJDL 9.7 Ki 3
WFPXOWCKXUEKCA 9.7 IC50 16
WSSWOLULTYVMTE 9.7 Ki 3
GOIFCXRIFSYPFG 9.7 Ki 5
CUCYVGNNTAIIAN 9.6 Ki 4
VACJUKKURQMWHE 9.6 Ki 5
KVKWRJDNIJTMGN 9.6 IC50 16
YMMRGIIZANFGIG 9.6 Ki 6
FIXFKUDATBTRAZ 9.6 Ki 4
ZRKDDZBVSZLOFS 9.6 Ki 6
QKIWQBLNTSQOLY 9.6 Ki 6
WQYYZNGOTUCWQX 9.6 Ki 5
IQKMZIHHJYCEKH 9.6 Ki 5
JUNLOSOXNSBSNV 9.6 Ki 3
RYKBQSSZEXHGJL 9.6 Ki 5
YIGPWWJHDOXRHC 9.6 Ki 4
LCDOZBPYZHDFGO 9.5 Ki 5
MCLMDSQSSOOSRY 9.5 Ki 3
NIPWDBCEPCGPGH 9.5 Ki 3
WMBPDZBHEAETLZ 9.5 Ki 3
XXAHGANHKMWQKV 9.5 Ki 3
KYDURMHFWXCKMW 9.5 Ki 6
LDXAQEAQNGTFAB 9.5 Ki 4
UWXAQZGCSSYTJL 9.5 Ki 6
VYBPWFTWAKMZPZ 9.5 Ki 5
KWZFUKSTRXYXTQ 9.4 Ki 3
RUOVJURXWIHZPL 9.4 Ki 5
CMSKDYKEKYIJSD 9.4 Ki 5
FGOCJZANGVRDDB 9.4 Ki 3
RXMRVZANJZUNED 9.4 Ki 3
PEBWTLIJBCZFOA 9.4 Ki 6
QXZGSQAJHBQSSV 9.4 Ki 4
RKXGEVUMNLOCDX 9.4 Ki 3
2D structure